Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with Target = 'Sensor protein kinase WalK' Sort by
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataIC50: 7.19E+3nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSensor protein kinase WalK(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453880(CHEMBL3343945)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of recombinant Staphylococcus epidermidis ATCC 35984 N-terminal GB1-tagged YycG expressed in Escherichia coli BL21 (DE3) preincubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSensor protein kinase WalK(Staphylococcus epidermidis (strain ATCC 35984 / RP...)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453886(CHEMBL4215525)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of recombinant Staphylococcus epidermidis ATCC 35984 N-terminal GB1-tagged YycG expressed in Escherichia coli BL21 (DE3) preincubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM15759(4-[7-(4-fluorophenyl)-5H-pyrrolo[2,3-b]pyrazin-6-y...)
Affinity DataIC50: 9.33E+4nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM27434(11,13-dimethyl-8-thia-3,5,10-triazatricyclo[7.4.0....)
Affinity DataIC50: 9.55E+4nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSensor protein kinase WalK(Staphylococcus aureus subsp. aureus CN1)
Williams College

Curated by ChEMBL
LigandPNGBDBM50453879(CHEMBL4202687)
Affinity DataIC50: 2.12E+5nMAssay Description:Inhibition of Staphylococcus aureus DHp-catalytic domain PhoR autophosphorylation expressed in Escherichia coli RIL in presence of gamma-32P-ATP by S...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM18134(AMP.P[NH]P | 5-Adenylyl imidodiphosphate | ({[({[(...)
Affinity DataIC50: 2.28E+5nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSensor protein kinase WalK(Staphylococcus aureus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM153747(ROCHE screening, 65)
Affinity DataIC50: 8.83E+8nMAssay Description:Inhibition of Streptococcus pneumoniae VicK autophosphorylation using compound at non-aggregating concentration after 30 mins in presence of [gamma-3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed