Report error Found 22 Enz. Inhib. hit(s) with Target = 'Sarcoplasmic/endoplasmic reticulum calcium ATPase 2'
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 383nMAssay Description:Activation of SERCA2a in C57BL/6N mouse sarcoplasmic reticulum assessed as increase in calcium release measured for 10 mins in presence of ATP by NAD...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Activation of SERCA2a in human HEK293T cells endoplasmic reticulum assessed as increase in calcium release measured for 10 mins in presence of ATP by...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 1.09E+4nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 9.20E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 7.60E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 8.60E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 3.43E+4nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of SERCA2b in mouse testicular microsomesMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rat)
University of Chemistry and Technology Prague
Curated by ChEMBL
University of Chemistry and Technology Prague
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat cerebellar microsomes SERCA2b by enzyme-coupled methodMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Rat)
University of Chemistry and Technology Prague
Curated by ChEMBL
University of Chemistry and Technology Prague
Curated by ChEMBL
Affinity DataIC50: 6.72E+3nMAssay Description:Inhibition of Wistar rat heart SERCA2a after 1 hrMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataKi: 5.30E+4nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
