Compile Data Set for Download or QSAR
Report error Found 150 Enz. Inhib. hit(s) with Target = 'Sarcoplasmic/endoplasmic reticulum calcium ATPase 1'
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097525(CHEMBL3586099)
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097535(CHEMBL3125414)
Affinity DataKd:  3.15E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097547(CHEMBL3125413)
Affinity DataKd:  7.50E+3nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097548(CHEMBL3586098)
Affinity DataKd:  9.65E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097549(CHEMBL3586097)
Affinity DataKd:  1.03E+5nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097550(CHEMBL3125412)
Affinity DataKd:  3.21E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097551(CHEMBL3125420)
Affinity DataKd:  4.81E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097552(CHEMBL3125415)
Affinity DataKd:  2.23E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097553(CHEMBL3586096)
Affinity DataKd:  2.01E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097554(Casearborin D)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097555(CHEMBL3586095)
Affinity DataKd:  1.01E+4nMAssay Description:Binding affinity to rabbit skeletal muscle SERCA1a preincubated for 5 mins followed by Mg-ATP addition measured over 6 mins by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097556(CHEBI:81104 | Alisol B)
Affinity DataKd:  2.70E+4nMAssay Description:Binding affinity to rabbit hind leg muscle SERCA1a by pyruvate kinase and lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50097557(CHEMBL3586100)
Affinity DataKd:  5.00E+4nMAssay Description:Binding affinity to rabbit hind leg muscle SERCA1a by pyruvate kinase and lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326743((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326738((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431166(CHEMBL2332554)
Affinity DataKd:  13nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431167(CHEMBL2332553)
Affinity DataKd:  79nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431168(CHEMBL2332552)
Affinity DataKd:  20nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431169(CHEMBL2332551)
Affinity DataKd:  1.70nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431170(CHEMBL2332105)
Affinity DataKd:  9.40nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431171(CHEMBL2332104)
Affinity DataKd:  2.60nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431172(CHEMBL2332103)
Affinity DataKd:  55nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431173(CHEMBL2332102)
Affinity DataKd:  13nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431174(CHEMBL2332101)
Affinity DataKd:  8.5nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50431175(CHEMBL2332100)
Affinity DataKd:  11nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326742((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-3,3a,4-trih...)
Affinity DataKd:  10nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to SERCA1a in sarcoplasmic reticulum vesicles of rabbit skeletal muscle after 2.5 to 6 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326748((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165369(12-(4-Amino-4-carboxy-butyrylamino)-dodecanoic aci...)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326743((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165368(Dodecanedioic acid mono-((2S,3aR,4S,6S,6aR,7S,9bS)...)
Affinity DataIC50: 2.08nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326737((3S,3aR,4S,6S,6aR,7S,8S,9bS)-3,3a-dihydroxy-3,6,9-...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326751((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 3nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of rabbit skeletal muscle SERCA1 assessed as reduction in calcium uptake preincubated for 10 mins followed by ATP addition and measured af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326749((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 9nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326742((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-3,3a,4-trih...)
Affinity DataIC50: 10nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326746((3S,3aR,4S,6S,6aR,7S,8S,9bS)-3a-hydroxy-3,6,9-trim...)
Affinity DataIC50: 11.1nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326739((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataIC50: 15.6nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326738((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataIC50: 16nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326750((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-8-(2-(biphe...)
Affinity DataIC50: 18nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326745(Octanoic acid(2aS,5aS,7S,7aR,8S,9S,10bS,10cR)-7-bu...)
Affinity DataIC50: 19nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165366(Pentanedioic acid mono-((2S,3aR,4S,6S,6aR,7S,9bS)-...)
Affinity DataIC50: 19.8nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326735((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a,6...)
Affinity DataIC50: 20nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326736((3S,3aR,4S,6S,6aR,7S,8S,9bS)-3,3a,6-trihydroxy-3,6...)
Affinity DataIC50: 20nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326741((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-(2-(biphenyl-4-yl)a...)
Affinity DataIC50: 27nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326752((3S,3aR,4S,6S,6aR,7S,8S,9bS)-6-acetoxy-4-(butyrylo...)
Affinity DataIC50: 44nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326740((3S,3aR,4S,6S,6aR,7S,8S,9bS)-4-(butyryloxy)-3,3a-d...)
Affinity DataIC50: 70nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Rabbit)
Albert-Ludwigs-University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50326744(Octanoic acid(2aS,5aS,7S,7aR,8S,9S,10bS,10cR)-7,10...)
Affinity DataIC50: 70nMAssay Description:Inhibition of rabbit sarcoplasmic reticulum calcium ATPase by ATP regeneration assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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