Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with Target = 'Relaxin-3 receptor 2'
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558042(CHEMBL4760798)
Affinity DataEC50:  0.347nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558042(CHEMBL4760798)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558038(CHEMBL4798311)
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558038(CHEMBL4798311)
Affinity DataEC50:  0.513nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50581020(CHEMBL5094669)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50581018(CHEMBL5084331)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558038(CHEMBL4798311)
Affinity DataKi:  1.60nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558038(CHEMBL4798311)
Affinity DataKi:  1.60nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50581017(CHEMBL5081158)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human RXFP4 expressed in CHOK1 cells assessed as inhibition of forskolin-stimulated intracellular cAMP accumulation preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50581019(CHEMBL5089949)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558045(CHEMBL4779813)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558045(CHEMBL4779813)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50581010(CHEMBL5072593)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50382993(CHEMBL2030702)
Affinity DataIC50: 3.47nMAssay Description:Agonist activity at RXFP4 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50581016(CHEMBL5083969)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50526407(CHEMBL4470544)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human RXFP4 expressed in CHOK1 cells assessed as inhibition of forskolin-stimulated intracellular cAMP accumulation preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558039(CHEMBL4752265)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558039(CHEMBL4752265)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558042(CHEMBL4760798)
Affinity DataKi:  5.5nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558042(CHEMBL4760798)
Affinity DataKi:  5.5nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50561918(CHEMBL4761849)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50561919(CHEMBL4781389)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547989(CHEMBL4747872)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50382992(CHEMBL2030701)
Affinity DataIC50: 7.94nMAssay Description:Agonist activity at RXFP4 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547992(CHEMBL4754473)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547990(CHEMBL4799795)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50526409(CHEMBL4522365)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human RXFP4 expressed in CHOK1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding after 3 hrs by scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547991(CHEMBL4740938)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50561922(CHEMBL4799017)
Affinity DataEC50:  14nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50382991(CHEMBL2030700)
Affinity DataIC50: 14.1nMAssay Description:Agonist activity at RXFP4 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558043(CHEMBL4742346)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558043(CHEMBL4742346)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558040(CHEMBL4791094)
Affinity DataKi:  19nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50561920(CHEMBL4764969)
Affinity DataEC50:  19nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558040(CHEMBL4791094)
Affinity DataKi:  19nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547989(CHEMBL4747872)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547989(CHEMBL4747872)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558043(CHEMBL4742346)
Affinity DataKi:  22nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558043(CHEMBL4742346)
Affinity DataKi:  22nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558044(CHEMBL4796474)
Affinity DataKi:  23nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558044(CHEMBL4796474)
Affinity DataKi:  23nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547989(CHEMBL4747872)
Affinity DataKi:  30nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547989(CHEMBL4747872)
Affinity DataKi:  30nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558039(CHEMBL4752265)
Affinity DataKi:  33nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558039(CHEMBL4752265)
Affinity DataKi:  33nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558040(CHEMBL4791094)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50558040(CHEMBL4791094)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50547990(CHEMBL4799795)
Affinity DataKi:  35nMAssay Description:Competitive binding affinity to human RXFP4 receptor transfected in CHO-K1 cells in presence of europium-labeled Eu(A)-R3/I5 by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
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