Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with Target = 'Protein ultraspiracle'
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488441(CHEMBL2286428)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488516(CHEMBL2286743)
Affinity DataEC50:  1.05E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488533(CHEMBL2286746)
Affinity DataEC50:  2.57E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178990(CHEMBL2286425)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488536(CHEMBL2286749)
Affinity DataEC50:  1.07E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488532(CHEMBL2286750)
Affinity DataEC50:  7.24E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488531(CHEMBL2286751)
Affinity DataEC50:  3.72E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488508(CHEMBL2286946)
Affinity DataEC50:  7.08E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488530(CHEMBL2286718)
Affinity DataEC50:  9.33E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488514(CHEMBL2286720)
Affinity DataEC50:  1.55E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488458(CHEMBL2286427)
Affinity DataEC50:  9.77E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488475(CHEMBL2286422)
Affinity DataEC50:  3.39E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488486(CHEMBL2286726)
Affinity DataEC50:  6.61E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488528(CHEMBL2286728)
Affinity DataEC50:  1.12E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  6.61E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488461(CHEBI:38451 | Halofenozide)
Affinity DataEC50:  7.76E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488454(CHEMBL2286436)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488519(CHEMBL2286714)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488534(CHEMBL2286717)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488468(CHEMBL2286448)
Affinity DataEC50: <1.32E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488537(CHEMBL2286463)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster Kc cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488535(CHEMBL2286741)
Affinity DataEC50:  9.77E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488474(CHEMBL2286423)
Affinity DataEC50:  2.57E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488529(CHEMBL2286724)
Affinity DataEC50:  1.29E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488515(CHEMBL2286740)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488499(CHEMBL2228437)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488507(CHEMBL2286723)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50179088(CHEMBL2286725)
Affinity DataEC50:  1.07E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488521(CHEMBL2286709)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488538(CHEMBL2286462)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster Kc cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488467(CHEBI:38457 | RH-5849)
Affinity DataEC50:  1.82E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488512(CHEMBL2286706)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488520(CHEMBL2286711)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488467(CHEBI:38457 | RH-5849)
Affinity DataEC50:  3.72E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488494(CHEMBL2286736)
Affinity DataEC50:  7.24E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488479(CHEMBL2228435)
Affinity DataEC50:  8.51E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488517(CHEMBL2286738)
Affinity DataEC50:  9.12E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488443(CHEMBL2286420)
Affinity DataEC50:  3.39E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488515(CHEMBL2286740)
Affinity DataEC50:  1.20E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178982(CHEMBL2228438)
Affinity DataEC50:  6.61E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488490(CHEMBL2286729)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488473(CHEMBL2286426)
Affinity DataEC50:  6.92E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster Kc cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488500(CHEMBL2286737)
Affinity DataEC50:  8.13E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488499(CHEMBL2228437)
Affinity DataEC50:  1.20E+5nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488498(CHEMBL2286744)
Affinity DataEC50:  6.03E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488489(CHEMBL2286747)
Affinity DataEC50:  1.32E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488473(CHEMBL2286426)
Affinity DataEC50:  2.82E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488497(CHEMBL2286719)
Affinity DataEC50:  3.24E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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