Compile Data Set for Download or QSAR
Report error Found 168 Enz. Inhib. hit(s) with Target = 'Protein Tat'
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(Neamine derivative | CHEMBL349996)
Affinity DataKd:  30nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(Pyrene-1-carboxylic acid [(4R,5S,6S)-5-amino-6-((2...)
Affinity DataKd:  290nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097338(Neamine derivative | CHEMBL408877)
Affinity DataKd:  25nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50410416(CHEMBL196072)
Affinity DataKd:  1.80E+3nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50410417(CHEMBL371627)
Affinity DataKd:  7.70E+3nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50410418(CHEMBL194688)
Affinity DataKd:  7.41E+5nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50410419(CHEMBL364677)
Affinity DataKd:  9.52E+5nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50398244(CHEMBL609728)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50476285(CHEMBL609729)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524874(CHEMBL4549436)
Affinity DataEC50:  1.10E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524875(CHEMBL4439569)
Affinity DataEC50:  3.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524876(CHEMBL4561296)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524877(CHEMBL4541346)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524878(CHEMBL4583543)
Affinity DataEC50:  2.90E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293-FlpIn.RV cells harboring LTR driven CBG reporter co-expressing CMV driven CBR reporter assess...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524879(CHEMBL4531268)
Affinity DataEC50:  3.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524880(CHEMBL4450163)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524881(CHEMBL4464472)
Affinity DataEC50:  1.90E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524882(CHEMBL4465202)
Affinity DataEC50:  3.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524874(CHEMBL4549436)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataEC50:  2.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524883(CHEMBL4447567)
Affinity DataEC50:  2.30E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524884(CHEMBL1386792)
Affinity DataEC50:  6.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524885(CHEMBL4445198)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524886(CHEMBL4467303)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524887(CHEMBL4446565)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524888(CHEMBL4540359)
Affinity DataEC50:  1.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524889(CHEMBL4552693)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524882(CHEMBL4465202)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM29589(Panobinostat | Faridak | LBH-589B | LBH-589 | US10...)
Affinity DataEC50:  130nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataEC50:  8.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524888(CHEMBL4540359)
Affinity DataEC50:  2.20E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524890(CHEMBL4460170)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524891(CHEMBL4526214)
Affinity DataEC50:  800nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524892(CHEMBL4576878)
Affinity DataEC50:  3.00E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524887(CHEMBL4446565)
Affinity DataEC50:  900nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524893(CHEMBL4545696)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524894(CHEMBL4538496)
Affinity DataEC50:  1.10E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524895(CHEMBL4526607)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524896(CHEMBL4453396)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524897(CHEMBL4466564)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524898(CHEMBL4454101)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524899(CHEMBL4458012)
Affinity DataEC50:  2.80E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524900(CHEMBL4541304)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524901(CHEMBL4464671)
Affinity DataEC50:  1.30E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524902(CHEMBL4442612)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524903(CHEMBL4470014)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524904(CHEMBL1506392)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524905(CHEMBL4546726)
Affinity DataEC50:  8.00E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524906(CHEMBL4436830)
Affinity DataEC50:  2.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Tat(HIV-1)
University of Massachusetts Medical School

Curated by ChEMBL
LigandPNGBDBM50524907(CHEMBL4452854)
Affinity DataEC50: >4.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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