Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Protein Nef/Tyrosine-protein kinase HCK'
TargetProtein Nef/Tyrosine-protein kinase HCK(Human)
University of Pittsburgh

LigandPNGBDBM36545(diphenylfuropyrimidine-4-aminopropylfuran | DFP-4A...)
Affinity DataIC50: 2.00E+3nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Nef/Tyrosine-protein kinase HCK(Human)
University of Pittsburgh

LigandPNGBDBM14807(DFP-4AP | 3-({5,6-diphenylfuro[2,3-d]pyrimidin-4-y...)
Affinity DataIC50: 5.10E+3nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Nef/Tyrosine-protein kinase HCK(Human)
University of Pittsburgh

LigandPNGBDBM36544(Diphenylfuropyrimidine-4-aminobutanol | DFP-4AB)
Affinity DataIC50: 1.60E+4nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein Nef/Tyrosine-protein kinase HCK(Human)
University of Pittsburgh

LigandPNGBDBM14806(DFP-4A | 5,6-diphenylfuro[2,3-d]pyrimidin-4-amine ...)
Affinity DataIC50: 3.00E+4nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed