Compile Data Set for Download or QSAR
Report error Found 67 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-7' Sort by
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50010992(CHEMBL3259883)
Affinity DataEC50:  4.20E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50010987(CHEMBL3259880)
Affinity DataEC50:  1.54E+4nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007199(CHEMBL3237863)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007198(CHEMBL3237862)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007196(CHEMBL3237864)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007206(CHEMBL3237867)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007200(CHEMBL3237873)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007193(CHEMBL3237865)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007207(CHEMBL3237860)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007207(CHEMBL3237860)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007202(CHEMBL3237868)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 7nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007201(CHEMBL3237870)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007205(CHEMBL3237871)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007209(CHEMBL3237874)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007197(CHEMBL3237869)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50277889(CHEMBL451887 | CARFILZOMIB)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007208(CHEMBL3237861)
Affinity DataIC50: 29nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007208(CHEMBL3237861)
Affinity DataIC50: 29nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50277889(CHEMBL451887 | CARFILZOMIB)
Affinity DataIC50: 43nMAssay Description:Inhibition of human 20S proteasome beta2 subunit using Ac-RLR-AMC as substrate preincubated for 2 hrs followed by substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007206(CHEMBL3237867)
Affinity DataIC50: 46nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007204(CHEMBL3237872)
Affinity DataIC50: 54nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50: 76nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015247(CHEMBL3262766)
Affinity DataIC50: 110nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007196(CHEMBL3237864)
Affinity DataIC50: 120nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 120nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007197(CHEMBL3237869)
Affinity DataIC50: 130nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007198(CHEMBL3237862)
Affinity DataIC50: 140nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007199(CHEMBL3237863)
Affinity DataIC50: 150nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007200(CHEMBL3237873)
Affinity DataIC50: 170nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015246(CHEMBL3262765)
Affinity DataIC50: 170nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015242(CHEMBL3262758)
Affinity DataIC50: 190nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007201(CHEMBL3237870)
Affinity DataIC50: 210nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015240(CHEMBL3262756)
Affinity DataIC50: 220nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007202(CHEMBL3237868)
Affinity DataIC50: 250nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015239(CHEMBL3262755)
Affinity DataIC50: 340nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015236(CHEMBL3262752)
Affinity DataIC50: 340nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015241(CHEMBL3262757)
Affinity DataIC50: 360nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015238(CHEMBL3262754)
Affinity DataIC50: 380nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015237(CHEMBL3262753)
Affinity DataIC50: 440nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007204(CHEMBL3237872)
Affinity DataIC50: 500nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015244(CHEMBL3262762)
Affinity DataIC50: 630nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50015243(CHEMBL3262761)
Affinity DataIC50: 950nMAssay Description:Inhibition of chymotrypsin-like enzyme activity of purified human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate by fluorescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007205(CHEMBL3237871)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50007198(CHEMBL3237862)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50430990(BELACTOSIN A)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50430990(BELACTOSIN A)
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of chymotrypsin-like of human 20S proteasome using chromophoric Suc-LLVY-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetProteasome subunit beta type-7(Human)
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
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