Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-4'
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577133(CHEMBL4870115)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577131(CHEMBL4855915)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50577116(CHEMBL4872258)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50604328(CHEMBL5180795)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of 20S proteasome subunit beta-2c (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50604324(CHEMBL5183361)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of 20S proteasome subunit beta-2c (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProteasome subunit beta type-4(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50604305(CHEMBL5209480)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of 20S proteasome subunit beta-2c (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185644((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185624((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  7.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185646(Pam-YKF | CHEMBL207452)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185645((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185625(pAM-FKF | CHEMBL380390)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(Pam-YDL | CHEMBL210871)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185628((S)-2-{(S)-4-carboxy-2-[(S)-2-dodecanoylamino-3-(4...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-4(Baker's yeast)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185633((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  3.15E+5nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed