Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with Target = 'Protachykinin-1'
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50281563(physalaemin | CHEMBL414786 | pGlu-Ala-Asp-Pro-Asn-...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81942(Neurokinin alpha | NSC_55582 | NKA | CAS_55582 | S...)
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81942(Neurokinin alpha | NSC_55582 | NKA | CAS_55582 | S...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81942(Neurokinin alpha | NSC_55582 | NKA | CAS_55582 | S...)
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81942(Neurokinin alpha | NSC_55582 | NKA | CAS_55582 | S...)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50194558(CHEMBL373569 | ELEDOISIN)
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81943(CAS_45749 | NSC_45749 | kassinin)
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81943(CAS_45749 | NSC_45749 | kassinin)
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50194558(CHEMBL373569 | ELEDOISIN)
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81943(CAS_45749 | NSC_45749 | kassinin)
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50194558(CHEMBL373569 | ELEDOISIN)
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50194558(CHEMBL373569 | ELEDOISIN)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81944(NSC_5311312 | NKB | CAS_86933-75-7 | neuromedin K)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81944(NSC_5311312 | NKB | CAS_86933-75-7 | neuromedin K)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81944(NSC_5311312 | NKB | CAS_86933-75-7 | neuromedin K)
Affinity DataKi:  56nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81944(NSC_5311312 | NKB | CAS_86933-75-7 | neuromedin K)
Affinity DataKi:  80nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  112nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50281563(physalaemin | CHEMBL414786 | pGlu-Ala-Asp-Pro-Asn-...)
Affinity DataKi:  113nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataKi:  125nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Mouse)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50281563(physalaemin | CHEMBL414786 | pGlu-Ala-Asp-Pro-Asn-...)
Affinity DataKi:  175nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM84994(NSC_163091 | CAS_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM81483(CAS_1893-33-0 | NSC_4830 | PIPAMPERONE)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM35255(2-Chloro-11-(2-(dimethylamino)ethoxy)dibenzo(b,f)t...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50095890(2-[2-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50001786(1-[2-[4-[5-chloro-1-(4-fluorophenyl)-indol-3-yl]-1...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50048803(5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-et...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM26948(CHEMBL46516 | cid_3396 | FLUSPIRILENE | 8-[4,4-bis...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Human)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM22913(CHEMBL1237146 | CHEMBL498770 | {[3-(1H-imidazol-5-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50035057(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazine |...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81818(CHEMBL1909810 | NSC_1794 | CAS_1794 | HMA)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81819(NSC_108107 | CHEMBL212579 | CAS_1937-37-7 | Benzam...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50010685((+/-)-trans-10,11-dihydroxy-5,6,6a,7,8,12b-hexahyd...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProtachykinin-1(Rat)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM50010685((+/-)-trans-10,11-dihydroxy-5,6,6a,7,8,12b-hexahyd...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed