Compile Data Set for Download or QSAR
Report error Found 740 Enz. Inhib. hit(s) with Target = 'Prostacyclin receptor'
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM62356(US9422273, 12b)
Affinity DataEC50:  860nMpH: 7.4 T: 2°CAssay Description:Ca2+ signaling studies were performed using a FLIPR TETRA system (Molecular Devices, Sunnyvale, Calif., USA) in the 384-format. This is a high-throug...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM240744(US9422273, 12a)
Affinity DataEC50:  550nMpH: 7.4 T: 2°CAssay Description:Ca2+ signaling studies were performed using a FLIPR TETRA system (Molecular Devices, Sunnyvale, Calif., USA) in the 384-format. This is a high-throug...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM240745(US9422273, 12c)
Affinity DataEC50:  9.50E+3nMpH: 7.4 T: 2°CAssay Description:Ca2+ signaling studies were performed using a FLIPR TETRA system (Molecular Devices, Sunnyvale, Calif., USA) in the 384-format. This is a high-throug...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM240746(US9422273, 12d)
Affinity DataEC50:  1.00E+3nMpH: 7.4 T: 2°CAssay Description:Ca2+ signaling studies were performed using a FLIPR TETRA system (Molecular Devices, Sunnyvale, Calif., USA) in the 384-format. This is a high-throug...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM240747(US9422273, 12e)
Affinity DataEC50:  290nMpH: 7.4 T: 2°CAssay Description:Ca2+ signaling studies were performed using a FLIPR TETRA system (Molecular Devices, Sunnyvale, Calif., USA) in the 384-format. This is a high-throug...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50101823(4-(2-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50101832((E)-7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50101829(7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-pro...)
Affinity DataEC50:  25nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50101822(CHEMBL64804 | PGE2, 15-epi | (Z)-7-[(1R,2R,3R)-3-H...)
Affinity DataEC50:  260nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50101853((13E,15S)-11alpha,15-dihydroxy-9-oxoprost-13-en-1-...)
Affinity DataEC50:  1.80nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50101824(Butaprost (Methyl Ester) | BUTAPROST | CHEMBL43252...)
Affinity DataEC50:  37nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103390(CHEMBL3398234)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103391(CHEMBL3398233)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103392(CHEMBL3398232)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103393(CHEMBL3398231)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103397(CHEMBL3398237)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103396(CHEMBL3398236)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103395(CHEMBL3398235)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103416(CHEMBL3398230)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103394(CHEMBL3398229)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103404(CHEMBL3398228)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103413(CHEMBL3398227)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103418(CHEMBL3398226)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103422(CHEMBL3398225)
Affinity DataEC50:  86nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103412(CHEMBL3398224)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103411(CHEMBL3398223)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103410(CHEMBL3398222)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103409(CHEMBL3398221)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103408(CHEMBL3398220)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103407(CHEMBL3398219)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103406(CHEMBL3398218)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103423(CHEMBL3398217)
Affinity DataEC50:  114nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103431(CHEMBL3398216)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103405(CHEMBL3398215)
Affinity DataEC50:  8.5nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103436(CHEMBL3398214)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103437(CHEMBL3398213)
Affinity DataEC50:  1.72E+3nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103403(CHEMBL3398212)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103402(CHEMBL3398211)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103401(CHEMBL3398210)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103400(CHEMBL3398209)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103399(CHEMBL3398208)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103438(CHEMBL3398207)
Affinity DataEC50:  2.67E+3nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Human)
Allergan

US Patent
LigandPNGBDBM50103398(CHEMBL3398206)
Affinity DataEC50:  969nMAssay Description:Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50103398(CHEMBL3398206)
Affinity DataEC50:  2.19E+3nMAssay Description:Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50103438(CHEMBL3398207)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50103399(CHEMBL3398208)
Affinity DataEC50:  310nMAssay Description:Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50103400(CHEMBL3398209)
Affinity DataEC50:  370nMAssay Description:Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50103401(CHEMBL3398210)
Affinity DataEC50:  900nMAssay Description:Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50103402(CHEMBL3398211)
Affinity DataEC50:  360nMAssay Description:Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstacyclin receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50103403(CHEMBL3398212)
Affinity DataEC50:  350nMAssay Description:Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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