Compile Data Set for Download or QSAR
Report error Found 360 Enz. Inhib. hit(s) with Target = 'Prokineticin receptor 2'
TargetProkineticin receptor 2(Human)
Central South University

LigandPNGBDBM121129(US8722896, (+/-)-1-Benzyl-N-(9-chloro-3,4- dihydro...)
Affinity DataIC50: 102nMpH: 7.5 T: 2°CAssay Description:Briefly, Chinese hamster ovary cells stably expressing the photoprotein aequorin were transiently transfected with WT or respective mutant PKR2-expre...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121106(US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  0.206nM ΔG°:  -57.5kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121324(US8722896, (-)-(2R)-2-Methyl-3-((3- hydroxy)benzyl...)
Affinity DataKi:  0.280nM ΔG°:  -56.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121105(US8722896, (-)-(3R)-1-(Indol-7-ylmethyl)-N- (9-chl...)
Affinity DataKi:  0.514nM ΔG°:  -55.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121086(US8722896, (-)-(3R)-1-(3-Hydroxybenzyl)- N-(9-chlo...)
Affinity DataKi:  0.550nM ΔG°:  -55.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121068(US8722896, (-)-(3R)-1-(2-Methoxybenzyl)- N-(9-chlo...)
Affinity DataKi:  0.680nM ΔG°:  -54.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121116(US8722896, (-)-(3R)-N-(9-chloro-3,4- dihydro-2H-1,...)
Affinity DataKi:  0.710nM ΔG°:  -54.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121040(US8722896, (+/-)-2-Methyl-3-((2- methoxy)benzylami...)
Affinity DataKi:  0.720nM ΔG°:  -54.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121070(US8722896, (-)-(3R)-1-(2-Methoxybenzyl)- N-(9-fluo...)
Affinity DataKi:  0.810nM ΔG°:  -54.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121319(US8722896, (+/-)-2-Methyl-3-((3- acetoxy)benzylami...)
Affinity DataKi:  0.890nM ΔG°:  -53.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121324(US8722896, (-)-(2R)-2-Methyl-3-((3- hydroxy)benzyl...)
Affinity DataKi:  0.930nM ΔG°:  -53.6kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121088(US8722896, (-)-(3R)-1-(3-Methoxybenzyl)- N-(9-chlo...)
Affinity DataKi:  1.03nM ΔG°:  -53.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121156(US8722896, (+/-)-2-Methyl-3-(1-((2- methoxypyridin...)
Affinity DataKi:  1.06nM ΔG°:  -53.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121261(US8722896, (-)-(3R)-1-(N-methyl-indol-4- ylmethyl)...)
Affinity DataKi:  1.24nM ΔG°:  -52.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Human)
Central South University

LigandPNGBDBM463312((-)-(2R)-1-(benzimidazol-4- ylmethyl)-N-(9-chloro-...)
Affinity DataKi:  1.30nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121040(US8722896, (+/-)-2-Methyl-3-((2- methoxy)benzylami...)
Affinity DataKi:  1.35nM ΔG°:  -52.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121253(US8722896, (-)-(2R)-2-Methyl-3-(indol-7- ylmethyla...)
Affinity DataKi:  1.39nM ΔG°:  -52.6kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121042(US8722896, (+)-(2S)-2-Methyl-3- benzylmethylamino)...)
Affinity DataKi:  1.40nM ΔG°:  -52.6kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121202(US8722896, (-)-(2R)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  1.43nM ΔG°:  -52.5kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121202(US8722896, (-)-(2R)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  1.5nM ΔG°:  -52.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121231(US8722896, (+/-)-(3R)-2-Methyl-3-(indolin-4- ylmet...)
Affinity DataKi:  1.53nM ΔG°:  -52.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121202(US8722896, (-)-(2R)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  1.60nM ΔG°:  -52.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121041(US8722896, (-)-(2R)-2-Methyl-3-((4- fluoro)benzyla...)
Affinity DataKi:  1.62nM ΔG°:  -52.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121143(US8722896, (+/-)-2-Methyl-3-((2- hydroxybenzyl)met...)
Affinity DataKi:  1.62nM ΔG°:  -52.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121070(US8722896, (-)-(3R)-1-(2-Methoxybenzyl)- N-(9-fluo...)
Affinity DataKi:  1.70nM ΔG°:  -52.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Human)
Central South University

LigandPNGBDBM463307((-)-(3R)-1-(benzimidazol-4- ylmethyl)-N-(9-chloro-...)
Affinity DataKi:  1.70nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121086(US8722896, (-)-(3R)-1-(3-Hydroxybenzyl)- N-(9-chlo...)
Affinity DataKi:  1.76nM ΔG°:  -52.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121145(US8722896, (+/-)-2-Methyl-3-((2- methoxybenzyl)met...)
Affinity DataKi:  1.76nM ΔG°:  -52.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121143(US8722896, (+/-)-2-Methyl-3-((2- hydroxybenzyl)met...)
Affinity DataKi:  1.77nM ΔG°:  -52.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121156(US8722896, (+/-)-2-Methyl-3-(1-((2- methoxypyridin...)
Affinity DataKi:  1.82nM ΔG°:  -51.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121205(US8722896, (-)-(2R)-2-Methyl-3-(indol-7- ylmethyla...)
Affinity DataKi:  1.85nM ΔG°:  -51.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121307(US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  1.86nM ΔG°:  -51.8kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121053(US8722896, (-)-(3R)-1-(2,3- Dimethylbenzyl)-N-(9-c...)
Affinity DataKi:  1.89nM ΔG°:  -51.8kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Human)
Central South University

LigandPNGBDBM463306((-)-(2R)-1-(4-Fluoro-3- methoxybenzyl)-N-(9-chloro...)
Affinity DataKi:  1.90nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121290(US8722896, (+/-)-(3R)-4-(Indol-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  1.94nM ΔG°:  -51.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Human)
Central South University

LigandPNGBDBM463309((+-)-2-Methyl-3-(benzimidazol- 4-ylmethylamino)-N-...)
Affinity DataKi:  2.10nMAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121262(US8722896, (-)-(3R)-1-(Indolin-4-ylmethyl)- N-(9-c...)
Affinity DataKi:  2.22nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121157(US8722896, (-)-(2R)-2-Methyl-3-(2,3- dihydro-1-ben...)
Affinity DataKi:  2.28nM ΔG°:  -51.3kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121157(US8722896, (-)-(2R)-2-Methyl-3-(2,3- dihydro-1-ben...)
Affinity DataKi:  2.38nM ΔG°:  -51.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121157(US8722896, (-)-(2R)-2-Methyl-3-(2,3- dihydro-1-ben...)
Affinity DataKi:  2.38nM ΔG°:  -51.2kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121104(US8722896, (-)-(3R)-1-(Indol-4-ylmethyl)-N- (9-chl...)
Affinity DataKi:  2.5nM ΔG°:  -51.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121291(US8722896, (+/-)-(3R)-4-(N-methyl-indol-4- ylmethy...)
Affinity DataKi:  2.5nM ΔG°:  -51.1kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121275(US8722896, (+/-)-4-(Indol-4-ylmethyl)-N-(9- chloro...)
Affinity DataKi:  2.60nM ΔG°:  -51.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121202(US8722896, (-)-(2R)-2-Methyl-3-(indol-4- ylmethyla...)
Affinity DataKi:  2.62nM ΔG°:  -51.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121259(US8722896, (-)-(3R)-1-(Indolin-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  2.62nM ΔG°:  -51.0kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121277(US8722896, (+/-)-4-(Indolin-4-ylmethyl)-N-(9- chlo...)
Affinity DataKi:  2.64nM ΔG°:  -50.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121111(US8722896, (-)-(3R)-1-Benzyl-N-(9-chloro- 3,4-dihy...)
Affinity DataKi:  2.66nM ΔG°:  -50.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121066(US8722896, (-)-(3R)-1-(2-Methoxybenzyl)- N-(3,4-di...)
Affinity DataKi:  2.67nM ΔG°:  -50.9kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121107(US8722896, (-)-(3R)-1-(Indolin-7-ylmethyl)- N-(9-c...)
Affinity DataKi:  2.87nM ΔG°:  -50.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProkineticin receptor 2(Chinese hamster)
The Regents of The University of California

US Patent
LigandPNGBDBM121205(US8722896, (-)-(2R)-2-Methyl-3-(indol-7- ylmethyla...)
Affinity DataKi:  2.87nM ΔG°:  -50.7kJ/moleT: 2°CAssay Description:An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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