Compile Data Set for Download or QSAR
Report error Found 542 Enz. Inhib. hit(s) with Target = 'Programmed cell death protein 1'
TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50507498(CHEMBL4436009)
Affinity DataKd:  3.39E+3nMAssay Description:Binding affinity to human PD1 (34 to 150 residues) expressed in Escherichia coli BL21 (DE3) measured for 120 secs by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50507499(CHEMBL4458745)
Affinity DataKd:  3.14E+3nMAssay Description:Binding affinity to human PD1 (34 to 150 residues) expressed in Escherichia coli BL21 (DE3) measured for 120 secs by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50507507(CHEMBL4544177)
Affinity DataKd:  3.13E+3nMAssay Description:Binding affinity to human PD1 (34 to 150 residues) expressed in Escherichia coli BL21 (DE3) measured for 120 secs by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50507508(CHEMBL4583803)
Affinity DataKd:  1.38E+3nMAssay Description:Binding affinity to human PD1 (34 to 150 residues) expressed in Escherichia coli BL21 (DE3) measured for 120 secs by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50546617(CHEMBL4793446)
Affinity DataKd:  1.66E+6nMAssay Description:Binding affinity to PD1 (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50580530(CHEMBL5092744)
Affinity DataKd:  3.30nMAssay Description:Binding affinity to human PD-1 assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM491057(US10975049, Example 26 | N-(4-(2-bromo-3-phenylben...)
Affinity DataIC50: 0.000500nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM507127(US11046675, Example 1006)
Affinity DataIC50: 2nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM581058(US11492375, Example 1120)
Affinity DataIC50: 4nMAssay Description:The ability of the macrocyclic peptides of the present disclosure to bind to PD-L1 was investigated using a PD-1/PD-L1 Homogenous Time-Resolved Fluor...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436120(US10590105, Example 1012)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436124(US10590105, Example 1016)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436128(US10590105, Example 1019)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436130(US10590105, Example 1020)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436133(US10590105, Example 1021)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436141(US10590105, Example 1028)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436142(US10590105, Example 1029)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436148(US10590105, Example 1034)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436149(US10590105, Example 1035)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436150(US10590105, Example 1036)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436157(US10590105, Example 1041)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436158(US10590105, Example 2001)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436159(US10590105, Example 2002)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436161(US10590105, Example 2004)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436163(US10590105, Example 2005)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436166(US10590105, Example 2008)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436169(US10590105, Example 2012)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436170(US10590105, Example 2013)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436172(US10590105, Example 2015)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM436173(US10590105, Example 2016)
Affinity DataIC50: 5nMAssay Description:The interaction of PD-1 and PD-L1 can be assessed using soluble, purified preparations of the extracellular domains of the two proteins. The PD-1 and...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482302(US10919852, Compound TABLE 1.1 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482303(US10919852, Compound TABLE 1.2 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482304(US10919852, Compound TABLE 1.3 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482305(US10919852, Compound TABLE 1.4 | US10919852, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482306(US10919852, Compound TABLE 1.5 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482307(US10919852, Compound TABLE 1.6 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482308(US10919852, Compound TABLE 1.7 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482309(US10919852, Compound TABLE 1.8 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482310(US10919852, Compound TABLE 1.9 | US11708326, Compo...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482311(US10919852, Compound TABLE 1.10 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482312(US10919852, Compound TABLE 1.11 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482313(US10919852, Compound TABLE 1.12 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482314(US10919852, Compound TABLE 1.13 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482315(US10919852, Compound TABLE 1.14 | US10919852, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482315(US10919852, Compound TABLE 1.14 | US10919852, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482317(US10919852, Compound TABLE 1.16 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482318(US10919852, Compound TABLE 1.17 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482320(US10919852, Compound TABLE 1.19 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482321(US10919852, Compound TABLE 1.20 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482322(US10919852, Compound TABLE 1.21 | US10919852, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetProgrammed cell death protein 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM482323(US10919852, Compound TABLE 1.22 | US11708326, Comp...)
Affinity DataIC50: 5nMAssay Description:96 Well plates were coated with 1 g/mL of human PD-L1 (obtained from R&D) in PBS overnight at 4° C. The wells were then blocked with 2% BSA in PBS (W...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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