Compile Data Set for Download or QSAR
Report error Found 186 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 1'
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50067880(4-methoxy-7H-furo[3,2-g]chromen-7-one | 5-methoxyp...)
Affinity DataKd: >2.00E+5nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50067878(9-Methoxy-furo[3',2':4,5]benzo[1,2-b][1,4]oxazin-3...)
Affinity DataKd:  2.90E+5nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50067881(4,9-Diethoxy-furo[3,2-g]chromen-7-one | CHEMBL3429...)
Affinity DataKd:  1.67E+5nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50067879(5-Methoxymethyl-3-methyl-furo[3,2-g]chromen-7-one ...)
Affinity DataKd:  5.60E+4nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50182587(5-acetyl-4-(4'-chloro)benzyloxy-6-hydroxy-7-methox...)
Affinity DataEC50:  1.70E+3nMAssay Description:Effect on blockade of Kv1.1 channelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50182585(5-acetyl-7-(4'-bromo)benzyloxy-6-hydroxy-4-methoxy...)
Affinity DataEC50:  1.20E+3nMAssay Description:Effect on blockade of Kv1.1 channelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50182597(5-acetyl-4,7-benzyloxy-6-hydroxybenzofuran | CHEMB...)
Affinity DataEC50:  7.00E+3nMAssay Description:Effect on blockade of Kv1.1 channelMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50375409(CHEMBL408488)
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of Kvbeta-1-mediated inactivation of Kv1.1 channel expressed in xenopus oocytes by voltage clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50375408(CHEMBL259345)
Affinity DataEC50:  6.00E+3nMAssay Description:Inhibition of Kvbeta-1-mediated inactivation of Kv1.1 channel expressed in xenopus oocytes by voltage clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50378799(CORTISONE)
Affinity DataEC50:  4.60E+4nMAssay Description:Activation of KV1.1 expressed in Xenopus laevis oocytes coexpressing Kvbeta1 assessed as increase in steady state current normalized to initial inact...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50378799(CORTISONE)
Affinity DataEC50:  3.30E+4nMAssay Description:Activation of KV1.1 expressed in Xenopus laevis oocytes coexpressing Kvbeta1 W155A mutant assessed as increase in steady state current normalized to ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115508(CHEMBL3609227)
Affinity DataIC50: 0.00100nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115569(CHEMBL3609231)
Affinity DataIC50: 0.00100nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115589(CHEMBL3609232)
Affinity DataIC50: 0.00100nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115603(CHEMBL3609245)
Affinity DataIC50: 0.00100nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115776(CHEMBL3609037)
Affinity DataIC50: 0.00100nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115501(CHEMBL3609220)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115504(CHEMBL3609223)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115676(CHEMBL3609265)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115699(CHEMBL3609032)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115701(CHEMBL3609034)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115792(CHEMBL3609045)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115804(CHEMBL3609055)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115813(CHEMBL3609061)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115632(CHEMBL3609069)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115637(CHEMBL3609074)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115638(CHEMBL3609075)
Affinity DataIC50: 0.00200nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115494(CHEMBL3608993)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115495(CHEMBL3608994)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115498(CHEMBL3608997)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115590(CHEMBL3609233)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115610(CHEMBL3609251)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115626(CHEMBL3609260)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115789(CHEMBL3609042)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115790(CHEMBL3609043)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115799(CHEMBL3609049)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115814(CHEMBL3609062)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115702(CHEMBL3609065)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115631(CHEMBL3609068)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115705(CHEMBL3609078)
Affinity DataIC50: 0.00300nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115505(CHEMBL3609224)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115593(CHEMBL3609236)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115595(CHEMBL3609238)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115598(CHEMBL3609240)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115674(CHEMBL3609263)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115683(CHEMBL3609272)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115689(CHEMBL3609276)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115788(CHEMBL3609041)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115798(CHEMBL3609048)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50115812(CHEMBL3609060)
Affinity DataIC50: 0.00400nMAssay Description:Antagonist activity at human Kv1.1 expressed in HEK293 cells assessed as inhibition of potassium currents after 10 mins by IonWorks Quattro patch cla...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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