Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with Target = 'Polyamine oxidase 1'
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294105(N-{8-[8-(N'-Cyclopropylmethyl-guanidino)-octylamin...)
Affinity DataKi:  0.0800nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294107(1-(Guanidino)-17-(N1-(beta-methylallyl)guanidino)-...)
Affinity DataKi:  0.5nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294109(1-(Guanidino)-17-(N1-(propargyl)guanidino)-9-azahe...)
Affinity DataKi:  0.700nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294108(1-(Guanidino)-17-(N1-(benzyl)guanidino)-9-azahepta...)
Affinity DataKi:  1nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294106(1-(Guanidino)-17-(N1-(gamma-methylallyl)guanidino)...)
Affinity DataKi:  1.10nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294110(1,17-Bis(N1-gamma.gamma-dimethylallyl)guanidino-9-...)
Affinity DataKi:  1.70nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294104(N-(8-{8-[N'-(3-Methyl-but-2-enyl)-guanidino]-octyl...)
Affinity DataKi:  3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50032500(Iminoctadiene | 1,1'-(8,8'-azanediylbis(octane-8,1...)
Affinity DataKi:  7.5nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294112(N-(gamma,gamma-Dimethylallyl)-N-(5-aminopentyl)-gu...)
Affinity DataKi:  10nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294111(N-prenyl agmatine | N-(4-Amino-butyl)-N'-(3-methyl...)
Affinity DataKi:  15nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294113(N-(gamma,gamma-Dimethylallyl)-N-(6-aminohexyl)-gua...)
Affinity DataKi:  22nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294114(1-allyl-3-(4-aminobutyl)guanidine | CHEMBL541766)
Affinity DataKi:  130nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294095(1-(4-aminobutyl)-3-(prop-2-ynyl)guanidine | CHEMBL...)
Affinity DataKi:  250nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50129716(OCTANE 1,8-DIAMINE | Octane-1,8-diamine | 1,8-diam...)
Affinity DataKi:  300nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294094(1-(4-aminobutyl)-3-(4-fluorophenyl)guanidine | CHE...)
Affinity DataKi:  630nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294103(4-[N3-gamma,gamma-Dimethyallyl)guanidino]-1-guanid...)
Affinity DataKi:  700nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294100(N1-(5-Aminopentyl)-N3-(3-methoxybenzyl)guanidine b...)
Affinity DataKi:  1.15E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294102(N1-[3'-Aminopropyl)-3-aminopropyl]-N3-(gamma,gamma...)
Affinity DataKi:  1.21E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294096(N-(3-Methyl-but-2-enyl)-N'-{4-[N'-(3-methyl-but-2-...)
Affinity DataKi:  1.50E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294099(N1-(5-Aminopentyl)-N3[(E)-3-phenyl-2-propenyl]guan...)
Affinity DataKi:  1.53E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294097(N1-(5-Aminopentyl)-N3-(cyclohexylethyl)guanidine b...)
Affinity DataKi:  1.72E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294098(N1-(5-Aminopentyl)-N3-(cyclopropylmethyl)guanidine...)
Affinity DataKi:  2.58E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM85213(CHEMBL58343 | US8633208, Agmatine | NSC_199 | CAS_...)
Affinity DataKi:  3.00E+3nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPolyamine oxidase 1(Maize)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50294101(N1-Benzylamine-N3-(gamma,gamma-dimethylallyl)guani...)
Affinity DataKi:  1.80E+4nMpH: 6.5Assay Description:Inhibition of maize PAO at pH 6.5 by spectrophotometry-based Dixon plot methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed