Report error Found 284 Enz. Inhib. hit(s) with Target = 'Pituitary adenylate cyclase-activating polypeptide'
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 4.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 52.5nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 389nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 37.6nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 52.2nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 834nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 37.6nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 20.6nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 8.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 2.60nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 7.70nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 0.700nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 1.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 7.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 4.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 0.700nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 10.1nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 4.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 49.4nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 3.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 1.03E+3nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 2.48E+3nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 564nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 4.01E+3nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 2.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 5.60nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 174nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 6.80nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 5.10nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 538nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 20.8nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 7.40nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 39.8nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 9.60nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 462nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 17.3nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 8.75nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 0.800nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 15.2nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Human)
Institut National De La Recherche Scientifique
Curated by ChEMBL
Institut National De La Recherche Scientifique
Curated by ChEMBL
Affinity DataEC50: 2.90nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
