Compile Data Set for Download or QSAR
Report error Found 123 Enz. Inhib. hit(s) with Target = 'Phospholipase A2 group V'
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50601469(CHEMBL5172164)
Affinity DataIC50: 10nMAssay Description:Inhibition of human group V phospholipase A2 expressed in Escherichia coli BL21(DE3) cells incubated for 10 to 20 mins cells by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50601469(CHEMBL5172164)
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse group V phospholipase A2 incubated for 10 to 20 mins cells by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263002((2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-6,7-benz...)
Affinity DataIC50: 20nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263002((2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-6,7-benz...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055391(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-ind...)
Affinity DataIC50: 44nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055391(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-ind...)
Affinity DataIC50: 57nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50262842(Benzenesulfonyl-2-(3-(2-amino-2-oxoacetyl)-1-benzy...)
Affinity DataIC50: 60nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263000(2-(1-benzyl-2-ethyl-1H-6,7-benzoindol-4-yloxy)-N-(...)
Affinity DataIC50: 70nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50262842(Benzenesulfonyl-2-(3-(2-amino-2-oxoacetyl)-1-benzy...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50274336(1-{3-Dodecanoyl-2,4,6-trihydroxy-5-[7-hydroxy-2-(4...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366(Varespladib sodium | (3-Aminooxalyl-1-benzyl-2-eth...)
Affinity DataIC50: 124nMAssay Description:Inhibition of recombinant human sPLA2-5 expressed in Escherichia coli BL21(DE3) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263000(2-(1-benzyl-2-ethyl-1H-6,7-benzoindol-4-yloxy)-N-(...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 170nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50458608(CHEMBL4205008)
Affinity DataIC50: 180nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50458608(CHEMBL4205008)
Affinity DataIC50: 180nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50333788((S)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366(Varespladib sodium | (3-Aminooxalyl-1-benzyl-2-eth...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50186585(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-6-meth...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366(Varespladib sodium | (3-Aminooxalyl-1-benzyl-2-eth...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50458606(CHEMBL4205511)
Affinity DataIC50: 510nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50458612(CHEMBL4214052)
Affinity DataIC50: 510nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50274336(1-{3-Dodecanoyl-2,4,6-trihydroxy-5-[7-hydroxy-2-(4...)
Affinity DataIC50: 520nMAssay Description:Inhibition of mouse sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50274337(1-(3-Dodecanoyl-2,4,6-trihydroxy-5-methyl-phenyl)-...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human sPLA2 group 5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50206911((+/+)-1-O-decyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H...)
Affinity DataIC50: 550nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 620nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50206920((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50: 660nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50458609(CHEMBL4213094)
Affinity DataIC50: 720nMAssay Description:Inhibition of sPLA2-5 (unknown origin) using 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine as substrate pretreated for 20 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366(Varespladib sodium | (3-Aminooxalyl-1-benzyl-2-eth...)
Affinity DataIC50: 750nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50186585(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-6-meth...)
Affinity DataIC50: 750nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366(Varespladib sodium | (3-Aminooxalyl-1-benzyl-2-eth...)
Affinity DataIC50: 750nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055383(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-methyl-1Hind...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50186586(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2,6-dimethyl-1...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50186586(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2,6-dimethyl-1...)
Affinity DataIC50: 850nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50055383(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-methyl-1Hind...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant sPLA2 G5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50206910((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50591714(CHEMBL5200953)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human PLA2G5More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50149981(CHEMBL3769794)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human group 5 secreted phospholipase A2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50591712(CHEMBL5194852)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of human PLA2G5More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50333789((R)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human group 5 sPLA2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50591713(CHEMBL5207115)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of human PLA2G5More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263051(2-(1-(2-amino-2-oxoacetyl)-2-(isobutyl)-3-(ophenyl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263051(2-(1-(2-amino-2-oxoacetyl)-2-(isobutyl)-3-(ophenyl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263052(2-[3-Biphenyl-2-ylmethyl-2-ethyl-8-(2-oxo-propoxy)...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263052(2-[3-Biphenyl-2-ylmethyl-2-ethyl-8-(2-oxo-propoxy)...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263053(2-(3-Biphenyl-2-ylmethyl-2-ethyl-8-methoxy-indoliz...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50263053(2-(3-Biphenyl-2-ylmethyl-2-ethyl-8-methoxy-indoliz...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50262843(Benzenesulfonyl-2-(3-(2-amino-2-oxoacetyl)-1-benzy...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhospholipase A2 group V(Mouse)
Niddk

Curated by ChEMBL
LigandPNGBDBM50262843(Benzenesulfonyl-2-(3-(2-amino-2-oxoacetyl)-1-benzy...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mouse group2V phospholipase A2 fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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