Compile Data Set for Download or QSAR
Report error Found 851 Enz. Inhib. hit(s) with Target = 'Phenylethanolamine N-methyltransferase'
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50176889(anti-9-amino-6-(trifluoromethyl)benzonorbornene | ...)
Affinity DataKd:  4.40E+3nMAssay Description:Activity of human wild type PNMT assessed as phenylethanolamine methylationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50176887(phenylethanolamine | CHEMBL224526)
Affinity DataKd:  1.80E+5nMAssay Description:Activity of human wild type PNMT assessed as phenylethanolamine methylationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50176888(3-trifluoromethylphenylethanolamine | CHEMBL224618)
Affinity DataKd:  2.40E+3nMAssay Description:Activity of human wild type PNMT assessed as phenylethanolamine methylationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM28422((2S)-2-amino-4-({[(2S,3S,4R,5R)-5-(6-amino-9H-puri...)
Affinity DataKd:  4.80E+3nMAssay Description:Activity of human wild type PNMT assessed as phenylethanolamine methylationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PNMTMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibitory potency was measured against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50240934(3-(hydroxymethyl)-N-(3,3,3-trifluoropropyl)-1,2,3,...)
Affinity DataIC50: 28nMAssay Description:Inhibition of PNMTMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028902(7,8-dichloro-2-[2-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50: 80nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029108(6,7,8-Trichloro-1,2,3,4-tetrahydro-isoquinoline | ...)
Affinity DataIC50: 100nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyl-transferase inhibitory potencyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028908(7,8-dichloro-2-[4-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029107(8-Chloro-1,2,3,4-tetrahydro-isoquinoline | CHEMBL1...)
Affinity DataIC50: 200nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyl-transferase inhibitory potencyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029101(5,6,7,8-Tetrachloro-1,2,3,4-tetrahydro-isoquinolin...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory potency was measured against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029102(7-Chloro-1,2,3,4-tetrahydro-isoquinoline | CHEMBL1...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory potency was measured against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028903(7,8-dichloro-2-[3-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029099(5,7,8-Trichloro-1,2,3,4-tetrahydro-isoquinoline | ...)
Affinity DataIC50: 300nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyl-transferase inhibitory potencyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029106(2,3-Dichloro-benzylamine | CHEMBL13165)
Affinity DataIC50: 600nMAssay Description:In vitro inhibitory potency was measured against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028910(7,8-dichloro-2-[6-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028901(7,8-Dichloro-2-ethyl-1,2,3,4-tetrahydro-isoquinoli...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028909(2-(7,8-Dichloro-3,4-dihydro-1H-isoquinolin-2-yl)-e...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028911(7,8-dichloro-2-[8-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028914(7,8-dichloro-2-[7-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028913(7,8-Dichloro-2-propyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028801(Cyclononanecarbaldehyde | CHEMBL18486)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028808(Cyclononyl-trimethylsilanyloxy-acetonitrile | CHEM...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028814(2-Amino-1-cyclononyl-ethanol | CHEMBL278978)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028783(CHEMBL18686 | CHEMBL1204148 | 2-Amino-1-cyclooctyl...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028912(2-Benzyl-7,8-dichloro-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028802(Cycloheptyl-trimethylsilanyloxy-acetonitrile | CHE...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028805(2-Amino-1-cycloheptyl-ethanol | CHEMBL280477)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028809(1-Trimethylsilanyloxy-cycloundecanecarbonitrile | ...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028812(Aldehydes, 6 | CHEMBL277996 | Cycloheptanecarbalde...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028651(1-Aminomethyl-cycloundecanol | CHEMBL18707)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028783(CHEMBL18686 | CHEMBL1204148 | 2-Amino-1-cyclooctyl...)
Affinity DataIC50: 8.00E+3nMAssay Description:The compound was measured for the 50% inhibition of phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028794(2-Amino-1-cycloundecyl-ethanol | CHEMBL19170)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028835(Cycloundecyl-trimethylsilanyloxy-acetonitrile | CH...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028846(Cycloundecanecarbaldehyde | CHEMBL279363)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM12584((3-chlorophenyl)methanamine | CHEMBL12957 | 1-(3-C...)
Affinity DataIC50: 9.00E+3nMAssay Description:In vitro inhibitory potency was measured against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028906(7,8-dichloro-2-[5-(7,8-dichloro-1,2,3,4-tetrahydro...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50028785(CHEMBL1204147 | CHEMBL18970 | 2-Amino-1-cyclohexyl...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028785(CHEMBL1204147 | CHEMBL18970 | 2-Amino-1-cyclohexyl...)
Affinity DataIC50: 1.40E+4nMAssay Description:The compound was measured for the 50% inhibition of phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028800(1-Aminomethyl-cyclononanol | CHEMBL278410)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028838(1-Trimethylsilanyloxy-cyclononanecarbonitrile | CH...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028851(Cyclononanone | CHEMBL276087)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029104(2-Chloro-benzylamine | CHEMBL12712)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory potency was measured against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50029105(2-(3,4,-dichlorophenyl)ethylamine | 2-(3,4-Dichlor...)
Affinity DataIC50: 2.00E+4nMAssay Description:Dissociation constant(Ki) of compound was determined to measure Phenylethanolamine N-methyl-transferase inhibitory potencyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028836(2-Amino-1-cyclooct-1-enyl-ethanol | CHEMBL18481)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPhenylethanolamine N-methyltransferase(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50028905(7,8-Dichloro-2-(6-phenyl-hexyl)-1,2,3,4-tetrahydro...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibitory activity against human phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50028828(2-Amino-1-cyclohex-3-enyl-ethanol | CHEMBL18594)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibitory activity against phenylethanolamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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