Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with Target = 'Penicillin-binding protein 1A' Sort by
TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708175(US12173018, Example 103)
Affinity DataEC50:  2.65E+5nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708306(US12173018, Example 5)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708107(US12173018, Example 17)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708109(US12173018, Example 20)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708111(US12173018, Example 22)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708114(US12173018, Example 26)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708115(US12173018, Example 27)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708119(US12173018, Example 34)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708129(US12173018, Example 45)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708130(US12173018, Example 46)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708133(US12173018, Example 49)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708146(US12173018, Example 70)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708147(US12173018, Example 71)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708152(US12173018, Example 76)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708311(US12173018, Example 85)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708158(US12173018, Example 86)
Affinity DataEC50: <3.00E+4nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708171(US12173018, Example 99)
Affinity DataEC50:  2.65E+5nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708172(US12173018, Example 100)
Affinity DataEC50:  2.65E+5nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A()
Venatorx Pharmaceuticals

US Patent
LigandPNGBDBM708174(US12173018, Example 102)
Affinity DataEC50:  2.65E+5nMAssay Description:To establish assay conditions for competition binding, an enzyme titration/saturation binding experiment was initially performed. Bocillin-FL was pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
Go to US Patent

TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 2.36nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3413 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 4.71nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3665 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 5.98nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 2527 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 9.43nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 24 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 9.43nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 1076 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50350464(Amoxi-Inject | Amoxi-Tabs | Amoxicillin | AMOXICIL...)
Affinity DataIC50: 10.9nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 24 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50483324(CHEBI:51257 | Faropenem)
Affinity DataIC50: 14nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3243 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 14.1nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 2527 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 14.1nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3243 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 18.9nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3676 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50422689(640/359 | CEFUROXIME)
Affinity DataIC50: 23.6nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3009 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 23.9nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3243 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 23.9nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 24 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 26.9nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3009 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 26.9nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 1077 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50012177(CHEMBL3265226)
Affinity DataIC50: 30nMAssay Description:Displacement of fluorescent Bocillin FL from N-terminal His tagged Pseudomonas aeruginosa PAO1 PBP1a (residues 36 to 822) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50483324(CHEBI:51257 | Faropenem)
Affinity DataIC50: 31.5nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 24 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50483324(CHEBI:51257 | Faropenem)
Affinity DataIC50: 35nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3009 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 35.9nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3676 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50012181(CHEMBL3265225)
Affinity DataIC50: 46nMAssay Description:Displacement of fluorescent Bocillin FL from N-terminal His tagged Pseudomonas aeruginosa PAO1 PBP1a (residues 36 to 822) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50012180(CHEMBL3265224)
Affinity DataIC50: 46nMAssay Description:Displacement of fluorescent Bocillin FL from N-terminal His tagged Pseudomonas aeruginosa PAO1 PBP1a (residues 36 to 822) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50012179(CHEMBL3265221)
Affinity DataIC50: 46nMAssay Description:Displacement of fluorescent Bocillin FL from N-terminal His tagged Pseudomonas aeruginosa PAO1 PBP1a (residues 36 to 822) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50012178(CHEMBL3265220)
Affinity DataIC50: 46nMAssay Description:Displacement of fluorescent Bocillin FL from N-terminal His tagged Pseudomonas aeruginosa PAO1 PBP1a (residues 36 to 822) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50350464(Amoxi-Inject | Amoxi-Tabs | Amoxicillin | AMOXICIL...)
Affinity DataIC50: 46.5nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 1077 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 47.8nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 1076 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50483324(CHEBI:51257 | Faropenem)
Affinity DataIC50: 52.6nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 1076 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50483324(CHEBI:51257 | Faropenem)
Affinity DataIC50: 52.6nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 1077 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50483324(CHEBI:51257 | Faropenem)
Affinity DataIC50: 56.1nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3413 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50022787((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...)
Affinity DataIC50: 59.8nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 3413 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50012182(CHEMBL3265223)
Affinity DataIC50: 65nMAssay Description:Displacement of fluorescent Bocillin FL from N-terminal His tagged Pseudomonas aeruginosa PAO1 PBP1a (residues 36 to 822) expressed in Escherichia co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetPenicillin-binding protein 1A(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Hershey Medical Center

Curated by ChEMBL
LigandPNGBDBM50483324(CHEBI:51257 | Faropenem)
Affinity DataIC50: 80.6nMAssay Description:Displacement of Biocillin FL from Streptococcus pneumoniae 2527 PBP1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
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