Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 6'
TargetP2X purinoceptor 6(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118219(Bz-ATP | CHEMBL339386)
Affinity DataEC50:  2.50E+4nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  1.00E+3nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118232(ATP, 2-meS | CHEMBL336208 | 2-MeSATP)
Affinity DataEC50:  600nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataEC50:  1.10E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118217(PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER | ATPga...)
Affinity DataEC50:  1.30E+3nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50336799(Suramin hexasodium | Germanin | suramin | 8,8'-[Ca...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118221(alpha,beta-meATP | DIPHOSPHOMETHYLPHOSPHONIC ACID ...)
Affinity DataEC50: >8.00E+3nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85043(CHEMBL69234 | CAS_149017-66-3 | NSC_6093163 | PPAD...)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85043(CHEMBL69234 | CAS_149017-66-3 | NSC_6093163 | PPAD...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of inward ion current elicited by ATP at rat P2X6 receptor (mutant type)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2X6 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50415550(Ro-85 | CHEMBL599760)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2X6 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2X purinoceptor 6(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85043(CHEMBL69234 | CAS_149017-66-3 | NSC_6093163 | PPAD...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of inward ion current elicited by ATP at rat P2X6 receptor (wild type)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed