Compile Data Set for Download or QSAR
Report error Found 358 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 5 group A member 2'
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418299(CHEMBL1765926)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418300(CHEMBL1765941)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418301(CHEMBL1765928)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418302(CHEMBL1765929)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22385((3aS,6aR)-5-hexyl-N,4-diphenyl-1,2,3,3a,6,6a-hexah...)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418312(CHEMBL1765932)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418306(CHEMBL1765955)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418304(CHEMBL1765953)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418310(CHEMBL1765962)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418303(CHEMBL1765959)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418313(CHEMBL1765945)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418308(CHEMBL1765933)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418309(CHEMBL1765956)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418325(CHEMBL1765958)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418307(CHEMBL1765934)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418326(CHEMBL1765961)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418305(CHEMBL1765960)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418316(CHEMBL1765966)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22373(bicyclo[3.3.0]-oct-2-ene, 5a | (3aS,6aR)-5-[(4E)-o...)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418329(CHEMBL1765951)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418311(CHEMBL1765931)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418321(CHEMBL1765963)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418330(CHEMBL1765938)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418324(CHEMBL1765957)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418317(CHEMBL1765950)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418323(CHEMBL1765964)
Affinity DataEC50:  1.58E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418314(CHEMBL1765954)
Affinity DataEC50:  1.58E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418315(CHEMBL1765936)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418318(CHEMBL1765942)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418319(CHEMBL1765930)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50418320(CHEMBL1765927)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22373(bicyclo[3.3.0]-oct-2-ene, 5a | (3aS,6aR)-5-[(4E)-o...)
Affinity DataEC50:  430nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22374((3aS,6aR)-4-methyl-5-[(4E)-oct-4-en-4-yl]-N-phenyl...)
Affinity DataEC50:  90nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22375((3aS,6aR)-4-butyl-5-[(4E)-oct-4-en-4-yl]-N-phenyl-...)
Affinity DataEC50:  22nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22376((3aS,6aR)-4-cyclohexyl-5-[(4E)-oct-4-en-4-yl]-N-ph...)
Affinity DataEC50:  12nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22377((3aS,6aR)-4-(4-bromophenyl)-5-[(4E)-oct-4-en-4-yl]...)
Affinity DataEC50:  160nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22378((3aS,6aR)-4-(3-methoxyphenyl)-5-[(4E)-oct-4-en-4-y...)
Affinity DataEC50:  100nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22379((3aS,6aR)-4-(naphthalen-2-yl)-5-[(4E)-oct-4-en-4-y...)
Affinity DataEC50:  60nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22380((3aS,6aR)-5-[(3E)-hex-3-en-3-yl]-N,4-diphenyl-1,2,...)
Affinity DataEC50:  1.40E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22381((3aS,6aR)-5-[(6E)-dodec-6-en-6-yl]-N,4-diphenyl-1,...)
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22382((3aS,6aR)-5-(hexan-2-yl)-N,4-diphenyl-1,2,3,3a,6,6...)
Affinity DataEC50:  70nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22383((3aS,6aR)-5-(decan-2-yl)-N,4-diphenyl-1,2,3,3a,6,6...)
Affinity DataEC50:  320nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22384((3aS,6aR)-5-methyl-N,4-diphenyl-1,2,3,3a,6,6a-hexa...)
Affinity DataEC50:  2.10E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22385((3aS,6aR)-5-hexyl-N,4-diphenyl-1,2,3,3a,6,6a-hexah...)
Affinity DataEC50:  34nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22386((3aS,6aR)-5-cyclohexyl-N,4-diphenyl-1,2,3,3a,6,6a-...)
Affinity DataEC50:  230nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22387((3aS,6aR)-5-dodecyl-N,4-diphenyl-1,2,3,3a,6,6a-hex...)
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22388((3aS,6aR)-N,4,5-triphenyl-1,2,3,3a,6,6a-hexahydrop...)
Affinity DataEC50:  150nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22389((3aS,6aR)-N-(3-fluorophenyl)-5-hexyl-4-phenyl-1,2,...)
Affinity DataEC50:  330nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22390((3aS,6aR)-N-(4-chlorophenyl)-5-hexyl-4-phenyl-1,2,...)
Affinity DataEC50:  1.00E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 5 group A member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM22391((3aS,6aR)-N-(2,3-dimethylphenyl)-5-hexyl-4-phenyl-...)
Affinity DataEC50:  30nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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