Compile Data Set for Download or QSAR
Report error Found 217 Enz. Inhib. hit(s) with Target = 'Neuropeptide FF receptor 1'
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50029096(CHEMBL3361425)
Affinity DataEC50:  3.52E+3nMAssay Description:Antagonist activity at human NPFF1 receptor expressed in CHO cells assessed as reversal of NPVF-induced inhibition of intracellular cAMP accumulation...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50029097(CHEMBL3361433)
Affinity DataEC50:  2.60E+3nMAssay Description:Antagonist activity at human NPFF1 receptor expressed in CHO cells assessed as reversal of NPVF-induced inhibition of intracellular cAMP accumulation...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50029098(CHEMBL3361418)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human NPFF1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50029109(CHEMBL3361419)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human NPFF1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50029111(CHEMBL3360829)
Affinity DataEC50:  4.70E+3nMAssay Description:Antagonist activity at human NPFF1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced intracellular cAMP accumulation relati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50029138(CHEMBL3360830)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human NPFF1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50029336(CHEMBL3361416)
Affinity DataEC50:  2.20E+4nMAssay Description:Antagonist activity at human NPFF1 receptor expressed in CHO cells assessed as reversal of NPVF-induced inhibition of intracellular cAMP accumulation...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50082073(CHEMBL3422407)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human NPFF1R expressed in CHO cells assessed as effect on forskolin-induced cAMP accumulation after 15 mins by luminescence based...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50082074(CHEMBL3422408)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human NPFF1R expressed in CHO cells assessed as effect on forskolin-induced cAMP accumulation after 15 mins by luminescence based...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50082065(CHEMBL3422516)
Affinity DataEC50:  222nMAssay Description:Agonist activity at human NPFF1R expressed in CHO cells assessed as effect on forskolin-induced cAMP accumulation after 15 mins by luminescence based...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM86143(RFamide-related peptide 3 | L-Val-L-Pro-L-Asn-L-Le...)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50394976(CHEMBL2165922)
Affinity DataKd:  41.7nMAssay Description:Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50060728((R)-5-(diaminomethyleneamino)-2-(2,2-diphenylaceta...)
Affinity DataKd:  20.9nMAssay Description:Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50394978(CHEMBL573297)
Affinity DataEC50:  527nMAssay Description:Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50394977(CHEMBL583068)
Affinity DataEC50:  2.37E+3nMAssay Description:Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50394975(CHEMBL2165921)
Affinity DataEC50:  5.62E+3nMAssay Description:Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50394977(CHEMBL583068)
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50414850(CHEMBL575058)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50414852(CHEMBL573738)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50414853(CHEMBL572825)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50414854(CHEMBL574565)
Affinity DataEC50:  39.8nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50414855(CHEMBL573518)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50414856(CHEMBL573519)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human NPFF1 receptor expressed in cells assessed as beta-galactosidase levels after 5 daysMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataEC50:  158nMAssay Description:Agonist activity at NPFF1 receptor (unknown origin) expressed in HEK293A cells assessed as inhibition of forskolin-stimulated cAMP accumulation measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to human NPFFR1 expressed in green monkey COS-7 cell membranes by [125I]-1DMeNPFF radioligand based saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50:  4.70E+3nMAssay Description:Antagonist activity at human NPFFR1 expressed in CHO cells assessed as reversal of NPVF-induced inhibition of forskolin-stimulated cAMP accumulation ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565181(CHEMBL4783555)
Affinity DataEC50:  599nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK-293A cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated fo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  589nMAssay Description:Partial agonist activity at NPFFR1 (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565182(CHEMBL4797394)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human NPFFR1 expressed in CHO cells by [35S]-GTP S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565183(CHEMBL4790994)
Affinity DataEC50:  176nMAssay Description:Agonist activity at human NPFFR1 expressed in CHO cells by [35S]-GTP S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50565184(CHEMBL4799458)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat NPFFR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565185(CHEMBL4777535)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human NPFFR1 by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565186(CHEMBL4785076)
Affinity DataEC50:  251nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in mouse NIH3T3 cells by receptor selection and amplification technology assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565187(CHEMBL4794542)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in mouse NIH3T3 cells by receptor selection and amplification technology assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565186(CHEMBL4785076)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293T cells harboring EP2 incubated for 15 mins by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565188(CHEMBL4784123)
Affinity DataEC50:  1.58E+4nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293T cells harboring EP2 incubated for 15 mins by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50565187(CHEMBL4794542)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293T cells harboring EP2 incubated for 15 mins by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558724(CHEMBL4796596)
Affinity DataEC50:  973nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558728(CHEMBL4777803)
Affinity DataEC50:  301nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558729(CHEMBL4788431)
Affinity DataEC50:  54nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558730(CHEMBL4792870)
Affinity DataEC50:  881nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558731(CHEMBL4777999)
Affinity DataEC50:  289nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558732(CHEMBL4759079)
Affinity DataEC50:  661nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558733(CHEMBL4785222)
Affinity DataEC50:  3.20E+3nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558734(CHEMBL4755334)
Affinity DataEC50:  928nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  591nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558724(CHEMBL4796596)
Affinity DataEC50:  977nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558728(CHEMBL4777803)
Affinity DataEC50:  302nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
The University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50558729(CHEMBL4788431)
Affinity DataEC50:  54nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 30...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 217 total ) | Next | Last >>
Jump to: