Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit beta-4'
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50110258(2-(6-Chloro-pyridin-3-yl)-9-aza-bicyclo[4.2.1]non-...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50110262(2-Pyridazin-4-yl-9-aza-bicyclo[4.2.1]non-2-ene | C...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50110260(2-Pyridin-3-yl-9-aza-bicyclo[4.2.1]non-2-ene | 2-P...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50023330(Anatoxin-a | Anatoxin-A,(+) | CHEMBL25619 | 1-(9-a...)
Affinity DataKi:  19nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50110259(2-Pyrimidin-5-yl-9-aza-bicyclo[4.2.1]non-2-ene | C...)
Affinity DataKi:  20nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  73nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM86311(CAS_485-35-8 | NSC_22407 | Cytisine | Cytisine-(-)...)
Affinity DataKi:  176nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit beta-4(Rat)
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50110263(2-Pyrazin-2-yl-9-aza-bicyclo[4.2.1]non-2-ene | CHE...)
Affinity DataKi:  259nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed