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Report error Found 2570 Enz. Inhib. hit(s) with Target = 'NACHT, LRR and PYD domains-containing protein 3'
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467910(CHEMBL4288029)
Affinity DataEC50:  630nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467913(CHEMBL4278564)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467915(CHEMBL4277080)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467916(CHEMBL4286476)
Affinity DataEC50:  520nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467919(CHEMBL4276704)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467920(CHEMBL4280136)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467921(CHEMBL4285025)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467917(CHEMBL4279629)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467914(CHEMBL4290288)
Affinity DataEC50:  610nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467912(CHEMBL4293700)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467918(CHEMBL4284645)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50467911(CHEMBL4283103)
Affinity DataEC50:  860nMAssay Description:Agonist activity at human NLRP3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50565841(CHEMBL4795253)
Affinity DataKd:  8.80nMAssay Description:Binding affinity to biotinylated human recombinant NLRP3 PYD domain by biolayer interferometry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50565841(CHEMBL4795253)
Affinity DataKd:  1.72E+4nMAssay Description:Binding affinity to biotinylated human recombinant NLRP3 NACHT domain by biolayer interferometry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50575103(CHEMBL4849582)
Affinity DataKd:  263nMAssay Description:Binding affinity to His-GFP fused tagged NLRP3 (unknown origin) expressed in HEK293T incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50597920(CHEMBL5180041)
Affinity DataKd:  1.63E+6nMAssay Description:Binding affinity to recombinant human full length NLRP3 expressed in Sf9 insect cells assessed as dissociation constant incubated for 30 mins by MST ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50598211(CHEMBL5173327)
Affinity DataKd:  84nMAssay Description:Binding affinity to human recombinant full length NLRP3 transfected in HEK293F cells assessed as dissociation constant incubated for 40 mins by micro...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50605172(CHEMBL5202921)
Affinity DataKd:  213nMAssay Description:Binding affinity to GFP-fused NLRP3 (unknown origin) expressed in HEK293T cells by MST assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622941(CHEMBL5417338)
Affinity DataKd:  25nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622942(CHEMBL5400432)
Affinity DataKd:  24nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622943(CHEMBL5409713)
Affinity DataKd:  0.980nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622944(CHEMBL5402231)
Affinity DataKd:  3nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622945(CHEMBL5435765)
Affinity DataKd:  700nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622946(CHEMBL5423405)
Affinity DataKd:  480nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622947(CHEMBL5430191)
Affinity DataKd:  0.860nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50622948(CHEMBL5434916)
Affinity DataKd:  69nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50632375(CHEMBL5430841)
Affinity DataKd:  5.87E+3nMAssay Description:Binding affinity to CMS sensor chip immobilized His-SUMO-tagged mouse NLRP3 expressed in Escherichia coli assessed as dissociation constant by SPR an...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50629371(CHEMBL5439097)
Affinity DataKd:  110nMAssay Description:Binding affinity to human recombinant NLRP3 (1 to 1036 residues) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50155926(CHEMBL3183703)
Affinity DataKd:  38nMAssay Description:Binding affinity to human recombinant NLRP3 (1 to 1036 residues) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633948(CHEMBL5401377)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633949(CHEMBL5410023)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633950(CHEMBL5437671)
Affinity DataEC50:  860nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633951(CHEMBL5416324)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633952(CHEMBL5433991)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633953(CHEMBL5439901)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633954(CHEMBL5405612)
Affinity DataEC50:  1.40E+4nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633955(CHEMBL5424007)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633956(CHEMBL5394766)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633957(CHEMBL5422678)
Affinity DataEC50:  5.70E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633958(CHEMBL5410936)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633959(CHEMBL5411420)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633960(CHEMBL5423650)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633961(Bms-986299 | BMS-986299)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633962(CHEMBL5429684)
Affinity DataEC50:  760nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633963(CHEMBL5417661)
Affinity DataEC50:  8.30E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633964(CHEMBL5422429)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633965(CHEMBL5396315)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633966(CHEMBL5438041)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633967(CHEMBL5400556)
Affinity DataEC50:  6.80E+3nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50633968(CHEMBL5418076)
Affinity DataEC50:  730nMAssay Description:Agonist activity at NLRP3 in human THP-1 cells assessed as LPS-stimulated IL-18 release incubated for 24 hrsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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