Compile Data Set for Download or QSAR
Report error Found 3394 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4'
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM43821(4-(2-benzamidoethylamino)-1-piperidinecarboxylic a...)
Affinity DataEC50:  2.14E+4nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 mus...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM43822(ethyl 4-[2-[(2-methylbenzoyl)amino]ethylamino]pipe...)
Affinity DataEC50:  2.40E+5nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of novel allosteric modulators of the M1 mus...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50323691(CHEMBL1212994 | cid_714286 | 3-amino-N-(4-chlorobe...)
Affinity DataEC50:  0.000339nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48043(3-amino-N-[(4-methoxyphenyl)methyl]-4,6-dimethyl-2...)
Affinity DataEC50:  388nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(VU0152099-1 | 3-amino-N-(1,3-benzodioxol-5-ylmethy...)
Affinity DataEC50:  369nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50323693(cid_734373 | CHEMBL1212983 | 3-amino-N-benzyl-4,6-...)
Affinity DataEC50:  0.000693nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48045(VU0402471-1 | cid_44176127 | 3-azanyl-N-[(2-fluoro...)
Affinity DataEC50:  0.000873nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48046(3-amino-N-[(2-chlorophenyl)methyl]-4,6-dimethylthi...)
Affinity DataEC50:  0.00234nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48047(cid_24769768 | 3-azanyl-N-[(3-chlorophenyl)methyl]...)
Affinity DataEC50:  0.00903nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48048(3-azanyl-4,6-dimethyl-N-[(3-methylphenyl)methyl]th...)
Affinity DataEC50:  0.0102nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48049(VU0402475-1 | cid_44176129 | 3-azanyl-4,6-dimethyl...)
Affinity DataEC50:  0.00282nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48050(3-azanyl-4,6-dimethyl-N-(pyridin-3-ylmethyl)thieno...)
Affinity DataEC50:  0.00559nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48051(3-azanyl-4,6-dimethyl-N-[(4-methylphenyl)methyl]th...)
Affinity DataEC50:  0.00242nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50323690(CHEMBL1212992 | VU10008 | cid_16757564 | 3-amino-4...)
Affinity DataEC50:  0.00242nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48052(VU0402479-1 | 3-amino-N-[(4-bromophenyl)methyl]-4,...)
Affinity DataEC50:  0.00516nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48053(cid_44176131 | 3-azanyl-4,6-dimethyl-N-[[4-(triflu...)
Affinity DataEC50:  0.00506nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48054(cid_44176132 | 3-azanyl-N-[[2,5-bis(fluoranyl)phen...)
Affinity DataEC50:  0.00100nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48055(3-azanyl-N-[[3,4-bis(fluoranyl)phenyl]methyl]-4,6-...)
Affinity DataEC50:  0.00127nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48056(3-amino-N-[(2,3-difluorophenyl)methyl]-4,6-dimethy...)
Affinity DataEC50:  0.000973nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48057(VU0152117 | 3-azanyl-6-[3-(dimethylamino)propoxy]-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48058(cid_45142470 | 3-azanyl-6-[2-(dimethylamino)ethoxy...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48059(VU0152119 | 3-amino-N-[(4-methoxyphenyl)methyl]-4-...)
Affinity DataEC50:  6.47E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48060(cid_45142472 | 3-azanyl-N-[(4-methoxyphenyl)methyl...)
Affinity DataEC50:  8.24E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48061(cid_45142473 | 3-amino-N-[(4-methoxyphenyl)methyl]...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48062(3-azanyl-N-[(4-methoxyphenyl)methyl]-4-methyl-6-pr...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48063(3-amino-N-[(4-methoxyphenyl)methyl]-4-methyl-6-pro...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48064(3-amino-N-[(4-methoxyphenyl)methyl]-4-methyl-6-(py...)
Affinity DataEC50:  1.97E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48065(VU0152130 | cid_44626303 | 3-amino-N-[(4-methoxyph...)
Affinity DataEC50:  2.21E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48066(cid_44626304 | VU0152131 | 3-amino-N-[(4-methoxyph...)
Affinity DataEC50:  1.77E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48067(3-azanyl-N-[(4-methoxyphenyl)methyl]-4-methyl-6-pe...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48068(3-azanyl-6-[3-(dimethylamino)propoxy]-4-methyl-N-(...)
Affinity DataEC50:  2.58E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48069(3-amino-N-[(2,5-difluorophenyl)methyl]-6-[3-(dimet...)
Affinity DataEC50:  2.75E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48070(VU0359453 | 3-azanyl-4-methyl-6-(2-morpholin-4-yle...)
Affinity DataEC50:  7.42E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48071(VU0359454 | 3-amino-N-(3-methoxypropyl)-4-methyl-6...)
Affinity DataEC50:  6.25E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48072(3-azanyl-4-methyl-6-(2-morpholin-4-ylethoxy)-N-pro...)
Affinity DataEC50:  7.15E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48073(3-amino-N-tert-butyl-4-methyl-6-[2-(4-morpholinyl)...)
Affinity DataEC50:  8.73E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48074(VU0359479 | 3-amino-N-[(2,3-difluorophenyl)methyl]...)
Affinity DataEC50:  5.40E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48075(VU0359480 | 3-amino-N-[(2,5-difluorophenyl)methyl]...)
Affinity DataEC50:  1.00E+4nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48076(ML173 | 3-azanyl-N-[[2,3-bis(fluoranyl)phenyl]meth...)
Affinity DataEC50:  1.61E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48077(VU0359509 | cid_45142487 | 3-azanyl-N-[[2,5-bis(fl...)
Affinity DataEC50:  1.58E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48078(3-azanyl-4-methyl-6-(2-morpholin-4-ylethoxy)-N-phe...)
Affinity DataEC50:  5.81E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48043(3-amino-N-[(4-methoxyphenyl)methyl]-4,6-dimethyl-2...)
Affinity DataEC50:  429nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(VU0152099-1 | 3-amino-N-(1,3-benzodioxol-5-ylmethy...)
Affinity DataEC50:  403nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48064(3-amino-N-[(4-methoxyphenyl)methyl]-4-methyl-6-(py...)
Affinity DataEC50:  1.97E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48076(ML173 | 3-azanyl-N-[[2,3-bis(fluoranyl)phenyl]meth...)
Affinity DataEC50:  1.67E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48043(3-amino-N-[(4-methoxyphenyl)methyl]-4,6-dimethyl-2...)
Affinity DataEC50:  87.1nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(VU0152099-1 | 3-amino-N-(1,3-benzodioxol-5-ylmethy...)
Affinity DataEC50: <1.42E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48064(3-amino-N-[(4-methoxyphenyl)methyl]-4-methyl-6-(py...)
Affinity DataEC50:  100nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48073(3-amino-N-tert-butyl-4-methyl-6-[2-(4-morpholinyl)...)
Affinity DataEC50:  192nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48076(ML173 | 3-azanyl-N-[[2,3-bis(fluoranyl)phenyl]meth...)
Affinity DataEC50:  95.3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
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