Compile Data Set for Download or QSAR
Report error Found 566 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase kinase 2'
LigandPNGBDBM40571(SMR000012776 | cid_648831 | MLS000032547 | 3-amino...)
Affinity DataEC50:  3.40E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51792(Pentanedioic acid cyclopentyl-cyclopentylcarbamoyl...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM32035(MLS000080234 | SMR000040438 | cid_659413)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM32050(SMR000044769 | MLS000080844 | cid_663844)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM34178(MLS000083027 | SMR000046592 | cid_665493 | 6-(2,6-...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51793(4-acetyl-N-(4,5-dihydrothiazol-2-yl)-3,5-dimethyl-...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM37692(SMR000015718 | cid_774866 | N2-(4-aminophenyl)benz...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51794(SMR000016567 | cid_3237248 | MLS000089497 | 1-cycl...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM44448(N-[2-(2-methyl-1-indolyl)ethyl]benzamide | SMR0000...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51795(cid_1091576 | 1-(5-chlorothiophen-2-yl)sulfonyl-4-...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM47934(N-[2-(2-methyl-1-indolyl)ethyl]-2-thiophenecarboxa...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM48177(MLS000106138 | SMR000103108 | cid_3103803)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM47717(MLS000525596 | SMR000116070 | 5-Ethylamino-anthra[...)
Affinity DataEC50:  4.43E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51796(MLS000526292 | SMR000116766 | (5Z)-5-[(2Z)-2-(3-et...)
Affinity DataEC50:  3.35E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51797(N-[2-(3-methylphenyl)-1,3-bis(oxidanylidene)isoind...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM43248(SMR000114403 | MLS000547610 | cid_1588252 | 5-[2-(...)
Affinity DataEC50:  3.22E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51798(SMR000127110 | cid_2136935 | MLS000530112 | 3-(4-f...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51799(MLS000518964 | 4-bromanyl-N-[5-(4-bromophenyl)imin...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51800(4-(1H-indol-3-yl)-N-methyl-2-thiazolamine | SMR000...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM43211(6-(4-Methoxy-phenyl)-2-piperazin-1-yl-pyrimidine-4...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM50056938(NSC-66209 | cid_72721 | CHEMBL175266 | 2,6,7-Trihy...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM39739(5-bromo-3-[2-[[(3Z)-2-(4-morpholinyl)-3-(phenylmet...)
Affinity DataEC50:  2.07E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51801(cid_11948850 | SMR000160726 | 4-[[4-[(2,4-dichloro...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM44965(cid_11948870 | 5-acetyloxy-6-bromo-2-[(carbamimido...)
Affinity DataEC50:  1.03E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51802(cid_6106925 | 4-({1-[3-(1H-imidazol-1-yl)propyl]-5...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51803(MLS000558753 | N-[(1E,3E)-4-(3-ethyl-1,3-benzothia...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51804(MLS000551916 | (3Z)-5-(4-ethoxyphenyl)-3-(3-pyridi...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM39775(SMR000174254 | MLS000557712 | 5-[3-(4-Dimethylamin...)
Affinity DataEC50:  910nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51805(3-[(3-chloranyl-4-methoxy-phenyl)methyl]-6,7-dimet...)
Affinity DataEC50:  2.23E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51806(6,7-dimethoxy-3-(4-methoxybenzyl)-2-[(2-methylbenz...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51807(N-{4-[(2-fluorobenzyl)oxy]-3-methoxybenzyl}-2-(1H-...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51808(SMR000194069 | 2-[[4-[(2-chlorophenyl)methoxy]phen...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM46560(SMR000194367 | MLS000572408 | N''-{4-[(2,4...)
Affinity DataEC50:  2.66E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51809(SMR000218462 | N-[[2,7-bis[2-(diethylamino)ethoxy]...)
Affinity DataEC50:  5.52E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51810(4-Methoxymethyl-6-methyl-5-nitro-2-phenethylamino-...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51811(SMR000221456 | MLS000331991 | 5-(4-Chloro-phenyl)-...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM50999(5-Benzo[1,3]dioxol-5-yl-1-methanesulfonyl-3-phenyl...)
Affinity DataEC50:  970nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51812(cid_3124282 | N-[4-(3-carbazol-9-yl-2-hydroxypropo...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51813(SMR000175579 | 3-[(4-methoxy-3-nitrophenyl)methyls...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM32299(cid_12004742 | MLS000559792 | 3-(2-Hydroxy-ethyl)-...)
Affinity DataEC50:  510nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM48732(SMR000212939 | cid_11293258 | (1-hexadecylpyridin-...)
Affinity DataEC50:  8.61E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51814(MLS000588973 | 2-butyl-N-[dibutoxyphosphoryl-(4-fl...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51815(MLS000580370 | 1-{[4-(4-Fluoro-phenyl)-thiazol-2-y...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51816(SMR000237271 | MLS000696829 | cid_12005896 | N-(4-...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51817(MLS000724906 | 1-(4-methoxyphenyl)-5-oxo-N-[5-(2-p...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51818(N-(6-chloro-1,3-benzothiazol-2-yl)-N-[3-(dimethyla...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51819(N-[3-[[4-(2-hydroxyethyl)piperazin-1-yl]-pyridin-2...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51820(MLS000331573 | SMR000220700 | 3-Hydroxy-naphthalen...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM46293(SMR000269408 | [3-(4-ethylphenyl)-1-phenyl-1H-pyra...)
Affinity DataEC50:  5.27E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51821(4-(4-penten-2-ynyl)-4-(3-phenyl-2-propynyl)morphol...)
Affinity DataEC50:  3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
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