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Report error Found 272 Enz. Inhib. hit(s) with Target = 'Lysophosphatidic acid receptor 3'
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  263nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148350([3-((Z)-Octadec-9-enoylamino)-thiopropionyl]-phosp...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50074700(Phosphoric acid mono-[2-((Z)-octadec-9-enoylamino)...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148353((1-Hydroxy-3-octadec-9-enoylamino-1-phosphono-prop...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148354([1-Fluoro-3-((Z)-octadec-9-enoylamino)-propyl]-pho...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148349((3-Octadec-9-enoylamino-propionyl)-phosphonothioic...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148355([3-((Z)-Octadec-9-enoylamino)-propyl]-phosphonic a...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148352([1-Hydroxy-3-((Z)-octadec-9-enoylamino)-propyl]-ph...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148351([3-((Z)-Octadec-9-enoylamino)-propionyl]-phosphoni...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at human LPA3 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166111((E)-Octadec-9-enoic acid (R)-2-fluoro-3-phosphonoo...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166113(Hexadecanoic acid (R)-2-fluoro-3-phosphonooxy-prop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166112((E)-Octadec-9-enoic acid (R)-2,2-difluoro-1-phosph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166116(Hexadecanoic acid (R)-4-fluoro-2-hydroxy-4-phospho...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166117(Hexadecanoic acid (S)-2-fluoro-3-phosphonooxy-prop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166114((E)-Octadec-9-enoic acid (S)-3,3-difluoro-1-phosph...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166115(CHEMBL190876 | PALMITOYL)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166118(Hexadecanoic acid (R)-2,2-difluoro-1-phosphonooxym...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166119(Hexadecanoic acid (S)-3,3-difluoro-1-phosphonooxym...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50166120(Hexadecanoic acid (S)-4-fluoro-2-methoxy-4-phospho...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170844(Thiophosphoric acid (E)-octadec-9-enyl ester | CHE...)
Affinity DataEC50:  546nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170848(2-Hexadecanoylamino-3-phosphonooxy-propionic acid ...)
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176390((R)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosp...)
Affinity DataEC50:  3nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176400((R)-2,3-bis(octyloxy)propyl dihydrogen phosphate |...)
Affinity DataEC50:  164nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176399(octanoic acid (S)-2-octanoyloxy-3-thiophosphonooxy...)
Affinity DataEC50:  115nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Rat)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50177334(potassium O-(2-(6-(4-octylphenyl)hexyl)-1,3-dioxol...)
Affinity DataEC50:  692nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Rat)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50177332(potassium O-(2-(heptadec-9-enyl)-1,3-dioxolan-4-yl...)
Affinity DataEC50:  639nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Rat)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50177338(potassium (2-(heptadeca-9,12,15-trienyl)-1,3-dioxo...)
Affinity DataEC50:  7.59E+3nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Rat)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50177330(potassium O-((2S,4S)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  265nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Rat)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50177328(potassium O-((2S,4R)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  127nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Rat)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50177335(potassium O-((2R,4R)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  194nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Rat)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50177333(potassium O-((2R,4S)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  204nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50193516(1,1-difluoro-3(S)-hydroxyl-4-oleoyloxylbutane 1,3-...)
Affinity DataEC50: >7.03E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50271700(4-(4-(ethoxycarbonyl)styryl)benzenesulfonic acid |...)
Affinity DataEC50: >1.18E+4nMAssay Description:Agonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at LPA3 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50381022(CHEMBL2017139)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430007(CHEMBL2335051)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430008(CHEMBL2335050)
Affinity DataEC50:  0.390nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430009(CHEMBL2335049)
Affinity DataEC50:  0.360nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430010(CHEMBL2335047)
Affinity DataEC50:  0.370nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430011(CHEMBL153043)
Affinity DataEC50:  0.440nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430012(CHEMBL357053)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430013(CHEMBL364797)
Affinity DataEC50:  580nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50233165(CHEMBL1222042)
Affinity DataEC50:  290nMAssay Description:Agonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as increase in intracellular calcium level measured every 3...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50610650(CHEMBL5285905)
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA3 receptorMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50610651(CHEMBL5277897)
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA3 receptorMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetLysophosphatidic acid receptor 3(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50610652(CHEMBL5281669)
Affinity DataEC50: <50nMAssay Description:Antagonist activity at human LPA3 receptorMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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