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Report error Found 124 Enz. Inhib. hit(s) with Target = 'Lysine--tRNA ligase'
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390557(CHEMBL2069346)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.860nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390556(CHEMBL2069345)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50249539(5-((1S,2R)-2-aminocyclohexylamino)-7-(3,5-dimethox...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390568(CHEMBL2069358)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390561(CHEMBL2069350)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390560(CHEMBL2069349)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390563(CHEMBL2069352)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390564(CHEMBL2069353)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390566(CHEMBL2069355)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390567(CHEMBL2069357)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465346(CHEMBL4286991)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390569(CHEMBL2069359)
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390562(CHEMBL2069351)
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50249254(5-((1S,2R)-2-aminocyclohexylamino)-7-(3,5-dimethox...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390573(CHEMBL2069356)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50249253(5-(2-aminoethylamino)-7-(3,5-dimethoxyphenylamino)...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390571(CHEMBL2069360)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465342(CHEMBL4293812)
Affinity DataIC50: 11nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390552(CHEMBL2069341)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465348(CHEMBL4292650)
Affinity DataIC50: 22nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390555(CHEMBL2069344)
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390565(CHEMBL2069354)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataIC50: 28nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465345(18-Oxoferruginol | acs.jmedchem.1c00409_ST.768)
Affinity DataIC50: 34nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50126419(N*1*-[7-(4-Dimethylamino-phenyl)-[1,6]naphthyridin...)
Affinity DataIC50: 34nMAssay Description:Inhibition of SYKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50249319(CHEMBL471901 | 2-(2-aminoethylamino)-4-(3-(trifluo...)
Affinity DataIC50: 41nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390559(CHEMBL2069348)
Affinity DataIC50: 43nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465347(POMIFERIN A | CHEBI:52486)
Affinity DataIC50: 46nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465338(CHEMBL598566 | 15-Hydroxydehydroabietic Acid)
Affinity DataIC50: 49nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50263121(cis-5-(2-Aminocyclohexylamino)-7-(3,5-dimethoxyphe...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390558(CHEMBL2069347)
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50426528(CHEMBL2323633)
Affinity DataIC50: 65nMAssay Description:Inhibition of human Gst-tagged Syk expressed in sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50426527(CHEMBL2323632)
Affinity DataIC50: 71nMAssay Description:Inhibition of human Gst-tagged Syk expressed in sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50426530(CHEMBL2323635)
Affinity DataIC50: 71nMAssay Description:Inhibition of human Gst-tagged Syk expressed in sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50242740(Type II inhibitor, 14 | CHEMBL459850 | N-(3-(7-Ami...)
Affinity DataEC50:  71nMAssay Description:Inhibition of Syk by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50426525(CHEMBL2323631)
Affinity DataIC50: 79nMAssay Description:Inhibition of human Gst-tagged Syk expressed in sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50263119(cis-5-(2-Aminocyclohexylamino)-7-(3,5-dimethoxyphe...)
Affinity DataIC50: 83nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465343(CHEMBL4279751)
Affinity DataIC50: 85nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390570(CHEMBL2069337)
Affinity DataIC50: 91nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465344(CHEMBL4294902)
Affinity DataIC50: 100nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465340(CHEMBL4278579)
Affinity DataIC50: 100nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465341(CHEMBL4289234)
Affinity DataIC50: 100nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50465339(CHEMBL4285076)
Affinity DataIC50: 100nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50390554(CHEMBL2069343)
Affinity DataIC50: 114nMAssay Description:Inhibition of human recombinant full-length Syk using poly-GT as substrate after 40 mins by radioactive filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50263120(cis-5-(2-Aminocyclohexylamino)-7-(3,5-dimethoxyphe...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Csir-National Chemical Laboratory

Curated by ChEMBL
LigandPNGBDBM50434379(CLADOSPORIN)
Affinity DataIC50: 120nMAssay Description:Inhibition of Plasmodium falciparum KRS expressed in Escherichia coli BL21 using tRNA(Lys) as substrate after 45 mins in presence of L-lysine by AMP-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50510261(CHEMBL4590082)
Affinity DataIC50: 140nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetLysine--tRNA ligase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50263040(5-(2-Amino-2-methylpropylamino)-7-(3,5-dimethoxyph...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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