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Report error Found 101 Enz. Inhib. hit(s) with Target = 'Lipoprotein lipase'
TargetLipoprotein lipase(Bovine)
Ume£

Curated by ChEMBL
LigandPNGBDBM50500148(CHEMBL3746381)
Affinity DataEC50:  6.60E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Bovine)
Ume£

Curated by ChEMBL
LigandPNGBDBM50500149(CHEMBL3747367)
Affinity DataEC50:  5.00E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Bovine)
Ume£

Curated by ChEMBL
LigandPNGBDBM50500150(CHEMBL3746821)
Affinity DataEC50:  6.00E+3nMAssay Description:Induction of bovine LPL stabilization using intralipid as substrate preincubated for 10 mins with human recombinant ANGPTL4 followed by substrate add...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254432(1-(2-methyl-5-(morpholinosulfonyl)furan-3-yl)-3-ph...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254434(5-Methyl-4-(3-phenyl-ureido)-furan-2-sulfonic acid...)
Affinity DataIC50: 50nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM24567(Tetrahydrolipstatin | CHEMBL175247 | Xenical | (2S...)
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant human LPL expressed in COS7 cells using PED-A1 containing DMPG vesicles as substrate pretreated for 20 mins followed by sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254436(5-Methyl-4-(3-phenyl-ureido)-furan-2-sulfonic acid...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254290(1-(2-methyl-5-(piperidin-1-ylsulfonyl)furan-3-yl)-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254340(1-(4-chlorophenyl)-3-(2-methyl-5-(piperidin-1-ylsu...)
Affinity DataIC50: 130nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254339(1-(4-methoxyphenyl)-3-(2-methyl-5-(piperidin-1-yls...)
Affinity DataIC50: 130nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138739(4-tert-butyl-N-(4-(5-methoxy-2-oxo-1,3,4-oxadiazol...)
Affinity DataIC50: 200nMAssay Description:Compound was tested to inhibit lipoprotein lipase (LPL)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254341(1-(2-chlorophenyl)-3-(2-methyl-5-(piperidin-1-ylsu...)
Affinity DataIC50: 320nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254435(5-Methyl-4-(3-phenyl-ureido)-furan-2-sulfonic acid...)
Affinity DataIC50: 400nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254343((S)-1-(2-methyl-5-(piperidin-1-ylsulfonyl)furan-3-...)
Affinity DataIC50: 400nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254433(1-(2-methyl-5-(4-methylpiperazin-1-ylsulfonyl)fura...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM26134((4-nonylphenyl)boranediol | Phenylboronic Acid, 13)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364285(CHEMBL1952298)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50433472(CHEMBL2381069)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of human LPL expressed in HEK293 cells using PED-A1 as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254393(1-benzhydryl-3-(2-methyl-5-(piperidin-1-ylsulfonyl...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50444153(CHEMBL3093304)
Affinity DataIC50: 2.56E+3nMAssay Description:Inhibition of recombinant human lipoprotein lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364283(CHEMBL1952296)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50253974(1-phenyl-3-(5-(piperidin-1-ylsulfonyl)furan-3-yl)u...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364295(CHEMBL1952307)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364298(CHEMBL1952310)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364282(CHEMBL1952295)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50067895(Tolyl boronic acid | p-tolylboronic acid | CHEMBL1...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364281(CHEMBL1952294)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364284(CHEMBL1952297)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364297(CHEMBL1952309)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50138734(3-(3-Benzyloxy-phenyl)-5-ethoxy-3H-[1,3,4]oxadiazo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested to inhibit lipoprotein lipase (LPL)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50444145(CHEMBL3093405)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human lipoprotein lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364295(CHEMBL1952307)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50521226(CHEMBL4471545)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of recombinant human LPL expressed in COS7 cells using PED-A1 containing DMPG vesicles as substrate pretreated for 20 mins followed by sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364282(CHEMBL1952295)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364300(CHEMBL1952312)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364283(CHEMBL1952296)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364299(CHEMBL1952311)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364292(CHEMBL1949700)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364293(CHEMBL1952305)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364301(CHEMBL1952313)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50254396(1-methyl-1-(2-methyl-5-(piperidin-1-ylsulfonyl)fur...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of Lipoprotein lipase from adipose tissue of ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364291(CHEMBL1952304)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364281(CHEMBL1952294)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50444138(CHEMBL3093392)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human lipoprotein lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50444152(CHEMBL3093305)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human lipoprotein lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364290(CHEMBL1952303)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364301(CHEMBL1952313)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364289(CHEMBL1952302)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed using recombinant adenovirus using glycerol-tri[9,10(n)-3H]oleate after 1 hr by vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50067895(Tolyl boronic acid | p-tolylboronic acid | CHEMBL1...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLipoprotein lipase(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50364289(CHEMBL1952302)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human lipoprotein lipase expressed in HEK293 cells using bis-BD-PC and mono-BD-TG as substrate incubated for 10 mins prior to substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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