Compile Data Set for Download or QSAR
Report error Found 352 Enz. Inhib. hit(s) with Target = 'Leucine-rich repeat serine/threonine-protein kinase 2 [970-2527,G2019S]'
LigandPNGBDBM254918(US9675594, 1 | US9499542, 1)
Affinity DataEC50:  201nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM254919(US9675594, 2 | US9499542, 2)
Affinity DataEC50:  195nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254920(US9675594, 3 | US9499542, 3)
Affinity DataEC50:  252nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254921(US9675594, 4 | US9499542, 4)
Affinity DataEC50:  851nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254922(US9675594, 5 | US9499542, 5)
Affinity DataEC50:  1.31E+3nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254923(US9675594, 6 | US9499542, 6)
Affinity DataEC50:  650nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254924(US9675594, 7 | US9499542, 7)
Affinity DataEC50:  78nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254925(US9675594, 8 | US9499542, 8)
Affinity DataEC50:  288nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254926(US9675594, 9 | US9499542, 9)
Affinity DataEC50:  26nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254927(US9675594, 10 | US9499542, 10)
Affinity DataEC50:  154nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254928(US9675594, 11 | US9499542, 11)
Affinity DataEC50:  240nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254929(US9675594, 12 | US9499542, 12)
Affinity DataEC50:  17nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254930(US9675594, 13 | US9499542, 13)
Affinity DataEC50:  58nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254931(US9675594, 14 | US9499542, 14)
Affinity DataEC50:  2nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254932(US9675594, 15 | US9499542, 15)
Affinity DataEC50:  1nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254933(US9675594, 16 | US9499542, 16)
Affinity DataEC50:  164nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254934(US9675594, 17 | US9499542, 17)
Affinity DataEC50:  527nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254935(US9675594, 18 | US9499542, 18)
Affinity DataEC50:  509nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254936(US9675594, 19 | US9499542, 19)
Affinity DataEC50:  215nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254937(US9675594, 20 | US9499542, 20)
Affinity DataEC50:  50nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254938(US9675594, 21 | US9499542, 21)
Affinity DataEC50:  575nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254939(US9675594, 22 | US9499542, 22)
Affinity DataEC50:  37nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM254940(US9675594, 23 | US9499542, 23)
Affinity DataEC50:  108nMAssay Description:In the assay, 1 nM LRRK2 WT or 250 pM LRRK2 G2019S kinase is incubated with the test compound (typically at 0 to 30 μM) for 30 minutes before th...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257380(US9493440, 230)
Affinity DataIC50: 0.450nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257387(US9493440, T2)
Affinity DataIC50: 0.490nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257316(US9493440, 160)
Affinity DataIC50: 0.520nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257175(US9493440, 16)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257184(US9493440, 26 | BDBM257386)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257194(US9493440, 38)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257285(US9493440, 129)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257287(US9493440, 131)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257289(US9493440, 133)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257295(US9493440, 139)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257307(US9493440, 151)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257309(US9493440, 153)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257311(US9493440, 155)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257312(US9493440, 156)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257326(US9493440, 170)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257330(US9493440, 174)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257342(US9493440, 186)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257161(US9493440, 1 | BDBM257389)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257184(US9493440, 26 | BDBM257386)
Affinity DataIC50: 0.600nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257189(US9493440, 33 | BDBM257192)
Affinity DataIC50: 0.630nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257189(US9493440, 33 | BDBM257192)
Affinity DataIC50: 0.630nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257315(US9493440, 159)
Affinity DataIC50: 0.670nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257371(US9493440, 219)
Affinity DataIC50: 0.670nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257193(US9493440, 37)
Affinity DataIC50: 0.700nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257271(US9493440, 115)
Affinity DataIC50: 0.700nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257284(US9493440, 128)
Affinity DataIC50: 0.700nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM257286(US9493440, 130)
Affinity DataIC50: 0.700nMpH: 8.5 T: 2°CAssay Description:a) 400 nl of a 1:2.15 serial dilution of test compound (98 uM top assay concentration) is spotted via Labcyte Echo to certain wells in a 384 well bla...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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