Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Isoform Beta of cGMP-dependent protein kinase 1 [5-676,G306E]'
LigandPNGBDBM65501(Cyclic GMP analogs | 8-pCP-cGMP | cGMP)
Affinity DataEC50:  370nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM65502(2-amino-8-bromo-9-[(2R,4aR,6R,7R,7aS)-2,7-dihydrox...)
Affinity DataEC50:  206nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM65501(Cyclic GMP analogs | 8-pCP-cGMP | cGMP)
Affinity DataEC50:  249nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  18nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed