Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'Integrin beta-3' Sort by
TargetIntegrin beta-3/subunit alpha 2b(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50453875(CHEMBL1811964)
Affinity DataEC50:  1.66E+3nMAssay Description:Binding affinity to GP2b/3a in rat blood assessed as conformational change by measuring soluble GP2b/3a levels after 12 hrs by UV-spectrophotometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetIntegrin beta-3(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50453876(CHEMBL4212580)
Affinity DataEC50:  1.16E+3nMAssay Description:Binding affinity to GP2b/3a in rat blood assessed as conformational change by measuring soluble GP2b/3a levels after 12 hrs by UV-spectrophotometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetIntegrin beta-3(Mouse)
University of Bradford

Curated by ChEMBL
LigandPNGBDBM50083811(3-({1-[3-(1H-Imidazol-2-ylamino)-propyl]-1H-indazo...)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at mouse endothelial alpha2bbeta3 integrin receptor by cell adhesion assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetIntegrin beta-3(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50004058(N-(butylsulfonyl)-O-(4-piperidin-4-ylbutyl)-L-tyro...)
Affinity DataIC50: 130nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetIntegrin beta-3(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50004058(N-(butylsulfonyl)-O-(4-piperidin-4-ylbutyl)-L-tyro...)
Affinity DataIC50: 136nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetIntegrin beta-3(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50568659(CHEMBL4861415)
Affinity DataIC50: 603nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetIntegrin beta-3(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50568659(CHEMBL4861415)
Affinity DataIC50: 610nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetIntegrin beta-3(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50568658(CHEMBL4853717)
Affinity DataIC50: 890nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetIntegrin beta-3(Rat)
Capital Medical University

Curated by ChEMBL
LigandPNGBDBM50568658(CHEMBL4853717)
Affinity DataIC50: 897nMAssay Description:Inhibition of fibrinogen binding to rat platelet integrin alpha2b beta3 by ELISA based solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed