Compile Data Set for Download or QSAR
Report error Found 391 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase p300 [1287-1666]/Histone acetyltransferase type B catalytic subunit'
LigandPNGBDBM564163(US11414384, Example 75 Isomer 4)
Affinity DataIC50: 8.76nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM564302(US11414384, Example 102 Isomer 4)
Affinity DataIC50: 9.36nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564276(US11414384, Example 99 Isomer 2)
Affinity DataIC50: 15.6nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564582(US11414384, Example 156 Isomer 2)
Affinity DataIC50: 17nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564178(US11414384, Example 79 Isomer 2)
Affinity DataIC50: 17.1nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564131(US11414384, Example 71 Isomer 2)
Affinity DataIC50: 17.7nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564374(US11414384, Example 114 Isomer 2)
Affinity DataIC50: 19nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564098(US11414384, Example 69 Isomer 4)
Affinity DataIC50: 20.7nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564706(US11414384, Example 173 Isomer 2)
Affinity DataIC50: 21.1nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564118(US11414384, Example 70 Isomer 4)
Affinity DataIC50: 21.8nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564639(US11414384, Example 167 Isomer 1)
Affinity DataIC50: 23.2nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564539(US11414384, Example 146 Isomer 2)
Affinity DataIC50: 26nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564369(US11414384, Example 113 Isomer 2)
Affinity DataIC50: 28nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564629(US11414384, Example 166 Isomer 2)
Affinity DataIC50: 28.8nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564436(US11414384, Example 126 Isomer 2)
Affinity DataIC50: 36.2nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564733(US11414384, Example 174 Isomer 2)
Affinity DataIC50: 39nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50542046(CHEMBL4633516 | US11414384, Example 84 Isomer 2)
Affinity DataIC50: 41nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564608(US11414384, Example 163 Isomer 2)
Affinity DataIC50: 41.9nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564141(US11414384, Example 72 Isomer 2)
Affinity DataIC50: 42.4nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564418(US11414384, Example 121 Isomer 2 | US11414384, Exa...)
Affinity DataIC50: 44nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564742(US11414384, Example 175 Isomer 2)
Affinity DataIC50: 44nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564253(US11414384, Example 95 Isomer 2)
Affinity DataIC50: 46nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564655(US11414384, Example 168 Isomer 2)
Affinity DataIC50: 53.1nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564746(US11414384, Example 176 Isomer 1)
Affinity DataIC50: 53.8nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564274(US11414384, Example 98 Isomer 2)
Affinity DataIC50: 58.3nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564286(US11414384, Example 101 Isomer 2)
Affinity DataIC50: 59.2nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564259(US11414384, Example 96 Isomer 2)
Affinity DataIC50: 62nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564113(US11414384, Example 70 Isomer 2)
Affinity DataIC50: 64.3nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564588(US11414384, Example 157 Isomer 2)
Affinity DataIC50: 66nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564575(US11414384, Example 153 Isomer 2)
Affinity DataIC50: 79.8nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564020(US11414384, Example 64 Isomer 2)
Affinity DataIC50: 80nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564528(US11414384, Example 142 Isomer 2)
Affinity DataIC50: 81.6nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564418(US11414384, Example 121 Isomer 2 | US11414384, Exa...)
Affinity DataIC50: 82nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564683(US11414384, Example 169 Isomer 2 | US11414384, Exa...)
Affinity DataIC50: 87.1nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564599(US11414384, Example 161 Isomer 2)
Affinity DataIC50: 95.1nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564015(US11414384, Example 64 Isomer 1)
Affinity DataIC50: 97nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564565(US11414384, Example 151 Isomer 2)
Affinity DataIC50: 101nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50542049(CHEMBL4639768 | US11414384, Example 100 Isomer 2)
Affinity DataIC50: 116nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564306(US11414384, Example 103 Isomer 2)
Affinity DataIC50: 118nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564619(US11414384, Example 166 Isomer 1)
Affinity DataIC50: 123nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564237(US11414384, Example 91 Isomer 4)
Affinity DataIC50: 134nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564604(US11414384, Example 162 Isomer 2)
Affinity DataIC50: 135nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564366(US11414384, Example 112 Isomer 2)
Affinity DataIC50: 136nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564613(US11414384, Example 164 Isomer 2)
Affinity DataIC50: 140nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564148(US11414384, Example 74 Isomer 1)
Affinity DataIC50: 154nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564150(US11414384, Example 74 Isomer 2)
Affinity DataIC50: 160nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564240(US11414384, Example 92 Isomer 3)
Affinity DataIC50: 164nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564285(US11414384, Example 101 Isomer 1)
Affinity DataIC50: 166nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564408(US11414384, Example 120 Isomer 2)
Affinity DataIC50: 172nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM564258(US11414384, Example 96 Isomer 1)
Affinity DataIC50: 182nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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