Compile Data Set for Download or QSAR
Report error Found 1410 Enz. Inhib. hit(s) with Target = 'Histamine H2 receptor'
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000348(CHEMBL3228794)
Affinity DataEC50:  590nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000382(SK&F-92058 | CHEBI:6896 | METIAMIDE)
Affinity DataEC50:  1.10E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000385(CHEMBL3228793)
Affinity DataEC50:  2.30E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000391(CHEMBL3228792)
Affinity DataEC50:  3.20E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000405(CHEMBL92526 | CHEMBL3228819)
Affinity DataEC50:  4.30E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000408(CHEMBL3228806)
Affinity DataEC50:  4.00E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000411(CHEMBL3228809)
Affinity DataEC50:  4.60E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000443(CHEMBL280584 | CHEMBL3228799)
Affinity DataEC50:  5.30E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000444(CHEMBL282206 | CHEMBL3228808)
Affinity DataEC50:  5.50E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000952(CHEMBL3228791)
Affinity DataEC50:  9.50E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000953(CHEMBL3228807)
Affinity DataEC50:  1.10E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000954(CHEMBL3228820)
Affinity DataEC50:  1.40E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000955(CHEMBL3228795)
Affinity DataEC50:  1.60E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000956(CHEMBL3228818)
Affinity DataEC50:  1.90E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000957(CHEMBL3228796)
Affinity DataEC50:  1.90E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000958(CHEMBL3228800)
Affinity DataEC50:  2.70E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000959(CHEMBL3228801)
Affinity DataEC50:  3.50E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000960(CHEMBL3228814)
Affinity DataEC50:  3.70E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000961(CHEMBL3228802)
Affinity DataEC50:  5.00E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000962(CHEMBL3228816)
Affinity DataEC50:  7.70E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000963(CHEMBL3228805)
Affinity DataEC50:  9.10E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000964(CHEMBL3228804)
Affinity DataEC50:  1.60E+5nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50127601(2-(1H-Imidazol-4-yl)-cyclopropylamine | CHEMBL5938...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]tiotidineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50127602(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]tiotidineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50127603(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]tiotidineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50127610((1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclo...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]tiotidineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50127609(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]tiotidineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50127604(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]tiotidineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50127606(2-(1H-Imidazol-4-yl)-cyclopropylamine | CHEMBL2940...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H2 receptor using [3H]tiotidineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413499(UR-PI295 | CHEMBL465170)
Affinity DataEC50:  186nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413505(CHEMBL515428)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413497(UR-PI288 | CHEMBL443896)
Affinity DataEC50:  813nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413498(UR-PI294 | CHEMBL475621)
Affinity DataEC50:  302nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413506(UR-PI147 | CHEMBL474617)
Affinity DataEC50:  3.55E+3nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413507(UR-PI182 | CHEMBL475620)
Affinity DataEC50:  490nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413500(UR-PI287 | CHEMBL471724)
Affinity DataEC50:  110nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413501(SK&F-91486 | SK-91486 | CHEMBL325327)
Affinity DataEC50:  2.57E+3nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413508(CHEMBL474448)
Affinity DataEC50:  288nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413503(UR-PI141 | CHEMBL514641)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413502(UR-PI104 | CHEMBL474447)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50377986(UR-AK24 | CHEMBL483406)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413504(CHEMBL474449)
Affinity DataEC50:  955nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413500(UR-PI287 | CHEMBL471724)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50377986(UR-AK24 | CHEMBL483406)
Affinity DataEC50:  16nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413502(UR-PI104 | CHEMBL474447)
Affinity DataEC50:  182nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Guinea pig)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50413503(UR-PI141 | CHEMBL514641)
Affinity DataEC50:  78nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig atrium assessed as increase in heart rateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413499(UR-PI295 | CHEMBL465170)
Affinity DataEC50:  141nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413506(UR-PI147 | CHEMBL474617)
Affinity DataEC50:  347nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Human)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50413507(UR-PI182 | CHEMBL475620)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human H2 receptor expressed in insect Sf9 cells co-expressing GsalphaS fusion protein assessed as gamma[32P]GTP binding by liquid...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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