Affinity DataEC50: 2.00E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataEC50: 170nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 70nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+4nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 9.20E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 590nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+4nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 830nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 740nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 940nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 440nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 850nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Activation of human recombinant glucokinase by matrix assay in presence of glucoseMore data for this Ligand-Target Pair
Affinity DataKd: 440nMAssay Description:Binding affinity to recombinant wild-type human pancreatic glucokinase expressed in Escherichia coli K-12 at 11 uM by isothermal titration calorimetr...More data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity to recombinant wild-type human pancreatic glucokinase expressed in Escherichia coli K-12 at 100 uM by isothermal titration calorimet...More data for this Ligand-Target Pair
Affinity DataKd: 500nMAssay Description:Binding affinity to recombinant wild-type human pancreatic glucokinase expressed in Escherichia coli K-12 by isothermal titration calorimetry in pres...More data for this Ligand-Target Pair
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
Affinity DataAssay Description:The GK activity was assessed spectrometrically by a coupled reaction with glucose-6-phosphate dehydrogenase (G6PDH). Briefly, GK catalyzes glucose ph...More data for this Ligand-Target Pair
Affinity DataEC50: 67.1nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+4nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataEC50: 1.87E+3nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
Affinity DataEC50: 2.53E+3nMAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
