Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Heat shock protein 90, putative'
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
Universidad De Navarra

Curated by ChEMBL
LigandPNGBDBM50406805(CHEMBL585793 | GNF-Pf-4574)
Affinity DataKd:  27nMAssay Description:Binding affinity to Plasmodium falciparum HSP90 nucleotide binding domain by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
Universidad De Navarra

Curated by ChEMBL
LigandPNGBDBM50406806(CHEMBL598685 | GNF-Pf-4035 | SJ000111021)
Affinity DataKd:  7nMAssay Description:Binding affinity to Plasmodium falciparum HSP90 nucleotide binding domain by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
Universidad De Navarra

Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)
Affinity DataKd:  169nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
Universidad De Navarra

Curated by ChEMBL
LigandPNGBDBM50534392(CHEMBL4446324)
Affinity DataKd:  2.56E+4nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
Universidad De Navarra

Curated by ChEMBL
LigandPNGBDBM50406805(CHEMBL585793 | GNF-Pf-4574)
Affinity DataKd:  2.81E+4nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
Universidad De Navarra

Curated by ChEMBL
LigandPNGBDBM50628234(CHEMBL4803806)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of recombinant his-tagged Plasmodium falciparum Hsp90 GHKL domain expressed in Escherichia coli BL21 (DE3) cells by bis-ANS binding assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed