Compile Data Set for Download or QSAR
Report error Found 341 Enz. Inhib. hit(s) with Target = 'Guanine nucleotide-binding protein subunit alpha-15 [Y147C]/Metabotropic glutamate receptor 2'
LigandPNGBDBM222972(US9315518, 5-2 | US9315518, 2-7)
Affinity DataEC50:  16.0nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222967(US9315518, 2-8)
Affinity DataEC50:  28.1nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222968(US9315518, 2-9)
Affinity DataEC50:  100nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222969(US9315518, 2-16)
Affinity DataEC50:  64.1nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222970(US9315518, 2-22)
Affinity DataEC50:  56.1nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222971(US9315518, 2-34)
Affinity DataEC50:  22.8nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222972(US9315518, 5-2 | US9315518, 2-7)
Affinity DataEC50:  322nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222973(US9315518, 6-4)
Affinity DataEC50:  29.0nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222974(US9315518, 8-6)
Affinity DataEC50:  513nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222975(US9315518, 8-9)
Affinity DataEC50:  270nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222976(US9315518, 8-14)
Affinity DataEC50:  134nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222977(US9315518, 8-38)
Affinity DataEC50:  17.9nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222978(US9315518, 11-5)
Affinity DataEC50:  391nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222979(US9315518, 14-6)
Affinity DataEC50:  123nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222980(US9315518, 17-15)
Affinity DataEC50:  594nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222981(US9315518, 17-20)
Affinity DataEC50:  333nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222982(US9315518, 18-10)
Affinity DataEC50:  2.19E+3nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222983(US9315518, 18-42)
Affinity DataEC50:  986nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222984(US9315518, 18-200)
Affinity DataEC50:  43.2nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222985(US9315518, 19-4)
Affinity DataEC50:  951nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222986(US9315518, 19-62)
Affinity DataEC50:  116nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222987(US9315518, 24-7)
Affinity DataEC50:  48.5nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222988(US9315518, 24-20)
Affinity DataEC50:  177nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222989(US9315518, 25-5)
Affinity DataEC50:  359nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222990(US9315518, 34-3)
Affinity DataEC50:  14.4nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM222991(US9315518, 38-5)
Affinity DataEC50:  1.18E+3nMAssay Description:The compounds of the present invention may be tested in a fluorescence laser imaging plate reader (FLIPR) based assay. This assay is a common functio...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213143(US9278960, 8-50 | US9636337, 8-50)
Affinity DataIC50: 4nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM212882(US9278960, 2-29 | US9663506, Example 2-29)
Affinity DataIC50: 5nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213110(US9278960, 8-18 | US9278960, 8-17 | US9636337, 8-1...)
Affinity DataIC50: 5nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213110(US9278960, 8-18 | US9278960, 8-17 | US9636337, 8-1...)
Affinity DataIC50: 5nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213133(US9278960, 8-41 | US9278960, 8-40 | US9636337, 8-4...)
Affinity DataIC50: 5nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213144(US9278960, 8-51 | US9636337, 8-51)
Affinity DataIC50: 5nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213074(US9278960, 6-21 | US9663506, Example 6-21)
Affinity DataIC50: 6nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213104(US9278960, 8-11 | US9278960, 8-10)
Affinity DataIC50: 6nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213113(US9278960, 8-28 | US9278960, 8-27 | US9278960, 8-2...)
Affinity DataIC50: 6nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213122(US9278960, 8-29 | US9636337, 8-29)
Affinity DataIC50: 6nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213126(US9278960, 8-33 | US9636337, 8-33)
Affinity DataIC50: 6nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM212880(US9278960, 2-27 | US9663506, Example 2-27)
Affinity DataIC50: 7nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213078(US9278960, 6-25 | US9663506, Example 6-25)
Affinity DataIC50: 7nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213104(US9278960, 8-11 | US9278960, 8-10)
Affinity DataIC50: 7nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213108(US9278960, 8-15 | US9636337, 8-15)
Affinity DataIC50: 7nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213125(US9278960, 8-32 | US9636337, 8-32)
Affinity DataIC50: 7nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213128(US9278960, 8-35 | US9636337, 8-35)
Affinity DataIC50: 7nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM212892(US9278960, 2-39 | US9663506, Example 2-39)
Affinity DataIC50: 8nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213006(US9278960, 4-90 | US9663506, Example 4-90)
Affinity DataIC50: 8nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213007(US9278960, 4-91 | US9663506, Example 4-91)
Affinity DataIC50: 8nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213012(US9278960, 4-96 | US9663506, Example 4-96)
Affinity DataIC50: 8nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213051(US9278960, 4-135 | US9663506, Example 4-135)
Affinity DataIC50: 8nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213060(US9278960, 6-7 | US9663506, Example 6-7)
Affinity DataIC50: 8nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM213091(US9278960, 7-29 | US9636337, 7-29)
Affinity DataIC50: 8nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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