Compile Data Set for Download or QSAR
Report error Found 417 Enz. Inhib. hit(s) with Target = 'Growth factor receptor-bound protein 2'
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080831([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-cyclohexylc...)
Affinity DataKd:  30nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080834({4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-pho...)
Affinity DataKd:  60nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080833([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-hydrox...)
Affinity DataKd:  155nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080830([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-phosph...)
Affinity DataKd:  60nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080832([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-1-methyl-2-...)
Affinity DataKd:  3nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080835([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-hydrox...)
Affinity DataKd:  250nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080836(4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-phos...)
Affinity DataKd:  45nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50087242(Pro-Ser-pTyr-Val-Asn-Val-Gln-Asn | CHEMBL422705)
Affinity DataKd:  18nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50087243(Pro-Ser-F2Pmp-Val-Asn-Val-Gln-Asn | CHEMBL436789)
Affinity DataKd:  200nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50087244(Ac-Pro-Phe-pTyr-Val-Asn-Val-Pro-NH2 | CHEMBL237124...)
Affinity DataKd:  30nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50087245(Pro-Ser-Pmp-Val-Asn-Val-Gln-Asn | CHEMBL345170)
Affinity DataKd:  260nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50139762([(16R,20S)-18-((S)-Carbamoylmethyl)-14-(5-methyl-i...)
Affinity DataKd:  0.0750nMAssay Description:Binding affinity to SH2 domain of GRB2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50139762([(16R,20S)-18-((S)-Carbamoylmethyl)-14-(5-methyl-i...)
Affinity DataKd:  0.0930nMAssay Description:In vitro binding affinity for Grb2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50139764(5-Methylindolyl derivative | CHEMBL423988)
Affinity DataKd:  0.0750nMAssay Description:In vitro binding affinity for Grb2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50118687(N-{1-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-propylc...)
Affinity DataKd:  23.8nM Kon:  0.0991M-1s-1 Koff:  4.18E+6s-1Assay Description:Apparent dissociation constant for human growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161466((R)-N-(1-{(S)-2-Carbamoyl-1-[2-(7-nitro-benzo[1,2,...)
Affinity DataKd:  119nM Kon:  0.140M-1s-1 Koff:  1.18E+6s-1Assay Description:Apparent dissociation constant for human growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161188((S)-4-{4-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-pro...)
Affinity DataKd:  97.8nMAssay Description:In vitro binding affinity for growth factor receptor bound protein 2 SH2 domain from human breast cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161189((S)-4-{5-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-pro...)
Affinity DataKd:  2.28nMAssay Description:In vitro binding affinity for growth factor receptor bound protein 2 SH2 domain from human breast cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161190(Phosphoric acid mono-[(S)-4-(2-acetylamino-2-{2-[(...)
Affinity DataKd:  23.8nMAssay Description:In vitro binding affinity for growth factor receptor bound protein 2 SH2 domain from human breast cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161189((S)-4-{5-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-pro...)
Affinity DataKd:  0.0970nMAssay Description:In vitro binding affinity for growth factor receptor bound protein 2 SH2 domain from human breast cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161191((S)-4-{2-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-pro...)
Affinity DataKd:  14.8nMAssay Description:In vitro binding affinity for growth factor receptor bound protein 2 SH2 domain from human breast cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161189((S)-4-{5-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-pro...)
Affinity DataKd:  2.28nMAssay Description:In vitro binding affinity for growth factor receptor bound protein 2 SH2 domain from human breast cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50161189((S)-4-{5-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-pro...)
Affinity DataKd:  4.30nMAssay Description:In vitro binding affinity for growth factor receptor bound protein 2 SH2 domain from human breast cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50168312(2-{4-[(16R,20S)-18-((S)-Carbamoylmethyl)-9-carboxy...)
Affinity DataKd:  3.62nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50139762([(16R,20S)-18-((S)-Carbamoylmethyl)-14-(5-methyl-i...)
Affinity DataKd:  1.47nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50168315([(7S,14R,18S)-18-Carbamoylmethyl-14-(5-methyl-indo...)
Affinity DataKd: >1.00E+3nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50168317([(15R,20S)-10-[4-(Benzyl-hydroxy-phosphinoylmethyl...)
Affinity DataKd:  35.3nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50168316(N-{4-[(7S,14R,18S)-18-Carbamoylmethyl-9-carboxymet...)
Affinity DataKd:  67nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50168318([(15R,20S)-18-Carbamoylmethyl-10-[4-(hydroxy-methy...)
Affinity DataKd:  16.2nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50168314([(7S,14R,18S)-18-Carbamoylmethyl-10-(4-carboxymeth...)
Affinity DataKd:  33nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50168313([(7S,14R,18S)-18-Carbamoylmethyl-10-(4-hydroxy-phe...)
Affinity DataKd: >1.00E+3nMAssay Description:Dissociation constant value against growth factor receptor bound protein 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50193149(({4-[(5'R,11'S,24'R,30'S)-11',30'-bis(carbamoylmet...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Grb2-SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50193150(({4-[(5S,11S)-11-(carbamoylmethyl)-3,6,9,12-tetrao...)
Affinity DataKd:  230nMAssay Description:Binding affinity to Grb2-SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50193151(({4-[(5'S,11'S,24'S,30'S)-11',30'-bis(carbamoylmet...)
Affinity DataKd:  1.80nMAssay Description:Binding affinity to Grb2-SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50193153(({4-[(2S)-2-[(1-{[(1S)-2-carbamoyl-1-({3-[1-({[(1S...)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to Grb2-SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50193152((13S,20S)-4-((S)-3-(1-(((S)-4-amino-1,4-dioxo-1-(p...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Grb2-SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50193154(({4-[(5R,11S)-11-(carbamoylmethyl)-3,6,9,12-tetrao...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Grb2-SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50198876(Ac-VPPPVPPRRR-NH2 | CHEMBL390420)
Affinity DataKd:  3.67E+3nMAssay Description:Binding affinity to recombinant Grb2-SH3 domain by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50198878(H-VPPPVPPRRR-OH | CHEMBL437932)
Affinity DataKd:  3.82E+4nMAssay Description:Binding affinity to recombinant Grb2-SH3 domain by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50198879(H-VPPPP(CH3)PPRRR-OH | CHEMBL439045)
Affinity DataKd:  1.16E+4nMAssay Description:Binding affinity to recombinant Grb2-SH3 domain by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208562((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  2.14E+3nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208563((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  458nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208565((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  2.18E+3nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208564((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  36nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208566((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  27nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208568((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  202nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208567(4-((4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propylam...)
Affinity DataKd:  871nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208570((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  106nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208569((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  272nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50208571((R)-4-(4-(((S)-4-amino-1-(3-(naphthalen-2-yl)propy...)
Affinity DataKd:  320nMAssay Description:Binding affinity to Grb2-SH2 domain by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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