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Report error Found 777 Enz. Inhib. hit(s) with Target = 'Glycogen phosphorylase, liver form'
TargetGlycogen phosphorylase, liver form(Mouse)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50560998(CHEMBL4759496)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of mouse liver Glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135554(4-{3-[(4-Nitro-pyridine-2-carbonyl)-amino]-naphtha...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135558(4-{3-Fluoro-2-[(4-nitro-pyridine-2-carbonyl)-amino...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24393(2,3-dichloro-N-{1-[(2R)-2,3-dihydroxypropyl]-2-oxo...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activity of the test compounds against human recombinant glycogen phosphorylase a (GPa) was monitored using 96-well microplate format....More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135553(4-{3-[(4-Chloro-pyridine-2-carbonyl)-amino]-naphth...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135565(4-{3-[(4-Methoxy-pyridine-2-carbonyl)-amino]-napht...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133440(1-(4-Chloro-benzyl)-4-(2-chloro-phenyl)-6-methyl-1...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27730((2S,3R)-3-(tert-butoxy)-2-{[4-(4-methoxyphenyl)-2-...)
Affinity DataIC50: 3nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27747((2S,3R)-3-(tert-butoxy)-2-{[2-({[4-(cyclopropylmet...)
Affinity DataIC50: 3nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135562(4-{2-[(4-Nitro-pyridine-2-carbonyl)-amino]-phenoxy...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27743((2S,3R)-3-(tert-butoxy)-2-{[2-({[4-(cyclopropylmet...)
Affinity DataIC50: 4nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27745((2S,3R)-3-(tert-butoxy)-2-[(2-{[(2,6-dimethyl-4-pr...)
Affinity DataIC50: 4nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27746((2S,3R)-3-(tert-butoxy)-2-[(2-{[(2,6-dimethyl-4-pr...)
Affinity DataIC50: 4nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135557(4-{3-[(4-Ethyl-pyridine-2-carbonyl)-amino]-naphtha...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133438(4-(2-Chloro-phenyl)-1-(3,4-dimethoxy-benzyl)-6-met...)
Affinity DataIC50: 4nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133442(4-(2-Chloro-phenyl)-6-methyl-1-(3-nitro-benzyl)-1,...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50194411((S)-2,3-dichloro-N-(1-(dimethylamino)-1-oxo-3-phen...)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human liver GPa by multienzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50255975((S)-2-cyclohexyl-2-(3-(3-(2,6-dichloro-4-(trifluor...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human liver glycogen phosphorylase A by fluorescence intensity endpoint assay in presence of glucoseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256329(1-(3-(3-mesitylureido)-2-naphthamido)cyclooctaneca...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human liver glycogen phosphorylase A by fluorescence intensity endpoint assay in presence of glucoseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM39807(CP-526,423)
Affinity DataIC50: 6nMpH: 7.2 T: 2°CAssay Description:Human liver glycogen phsphorylase (HLGP) activity was measured in the direction of glycogen synthesis by the release of phosphate from glucose-1-phos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50149207(BIS[5-CHLORO-1H-INDOL-2-YL-CARBONYL-AMINOETHYL]-ET...)
Affinity DataIC50: 6nMAssay Description:Inhibition of glycogen phosphorylase a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50255977((S)-2-cyclohexyl-2-(3-(3-mesitylureido)-2-naphtham...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human liver glycogen phosphorylase A by fluorescence intensity endpoint assay in presence of glucoseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256669((2S,3R)-2-(3-(3-mesitylureido)-2-naphthamido)-3-(1...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human liver glycogen phosphorylase A by fluorescence plate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Mouse)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50149207(BIS[5-CHLORO-1H-INDOL-2-YL-CARBONYL-AMINOETHYL]-ET...)
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration against glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24385(2,3-dichloro-N-[1-(2-hydroxyethyl)-2-oxo-1,2,3,4-t...)
Affinity DataIC50: 7nMpH: 7.2 T: 2°CAssay Description:The inhibitory activity of the test compounds against human recombinant glycogen phosphorylase a (GPa) was monitored using 96-well microplate format....More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27726((2S,3R)-3-(tert-butoxy)-2-[(3-{[(2,4,6-trimethylph...)
Affinity DataIC50: 7nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27734((2S,3R)-3-(tert-butoxy)-2-{[4-(4-fluorophenyl)-2-{...)
Affinity DataIC50: 7nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27744((2S,3R)-3-(tert-butoxy)-2-{[4-(3,4-difluorophenyl)...)
Affinity DataIC50: 7nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27726((2S,3R)-3-(tert-butoxy)-2-[(3-{[(2,4,6-trimethylph...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human liver glycogen phosphorylase A by fluorescence plate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133443(4-(2-Chloro-phenyl)-1-ethyl-5-isobutylcarbamoyl-6-...)
Affinity DataIC50: 7.88nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27731((2S,3R)-3-(tert-butoxy)-2-{[4-(3-methoxyphenyl)-2-...)
Affinity DataIC50: 8nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133431(1-(3-Chloro-benzyl)-4-(2-chloro-phenyl)-6-methyl-1...)
Affinity DataIC50: 8nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135550(4-{2-[(4-Chloro-pyridine-2-carbonyl)-amino]-3-fluo...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against rat liver glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Mouse)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50135550(4-{2-[(4-Chloro-pyridine-2-carbonyl)-amino]-3-fluo...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against mouse liver glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50194415(2,3-dichloro-N-((1R,2R)-1-hydroxy-2,3-dihydro-1H-i...)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human liver GPa by multienzyme coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256573((S)-2-(3-(3-mesitylureido)-2-naphthamido)-5-methyl...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human liver glycogen phosphorylase A by fluorescence plate reader assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133444(4-(2-Chloro-phenyl)-1-ethyl-5-isopropylcarbamoyl-6...)
Affinity DataIC50: 9.10nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27729((2S,3R)-3-(tert-butoxy)-2-[(4-phenyl-2-{[(2,4,6-tr...)
Affinity DataIC50: 10nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM27742((2S,3R)-3-(tert-butoxy)-2-[(2-{[(2,6-dimethyl-4-pr...)
Affinity DataIC50: 10nMpH: 7.6 T: 2°CAssay Description:An enzymatic assay was developed to measure the response of the activated form of glycogen phosphorylase to small molecule compounds. The assay was t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135560(4-{3-[(4-Methyl-pyridine-2-carbonyl)-amino]-naphth...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135550(4-{2-[(4-Chloro-pyridine-2-carbonyl)-amino]-3-fluo...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50256169((S)-2-cyclohexyl-2-(3-(3-mesitylureido)-2-naphtham...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human liver glycogen phosphorylase A by fluorescence intensity endpoint assay in presence of glucoseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133429(5-Benzylcarbamoyl-4-(2-chloro-phenyl)-1-ethyl-6-me...)
Affinity DataIC50: 10.9nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135561(4-{3-Fluoro-2-[(4-methoxy-pyridine-2-carbonyl)-ami...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133430(1-Benzyl-4-(2-chloro-phenyl)-6-methyl-1,4-dihydro-...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM24399(2-chloro-N-[(3S)-1-[(2S)-2,3-dihydroxypropyl]-2-ox...)
Affinity DataIC50: 12nMAssay Description:The inhibitory activity of the test compounds against human recombinant glycogen phosphorylase a (GPa) was monitored using 96-well microplate format....More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135567(4-{3-[(4-Trifluoromethyl-pyridine-2-carbonyl)-amin...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50158278(5-Chloro-1H-indole-2-carboxylic acid {[(1,1-dioxo-...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50246785((2E,2'E)-N,N'-(Thiodiethane-2,1-diyl)bis[3-(3,4-di...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human liver glycogen phosphorylase a in presence of glucoseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50133433(4-(2-Chloro-phenyl)-1-ethyl-5-ethylcarbamoyl-6-met...)
Affinity DataIC50: 12.4nMAssay Description:In vitro inhibitory activity against human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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