Compile Data Set for Download or QSAR
Report error Found 2207 Enz. Inhib. hit(s) with Target = 'Glucose-dependent insulinotropic receptor'
LigandPNGBDBM50418004(CHEMBL2092727)
Affinity DataEC50:  44nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50418005(CHEMBL2092875)
Affinity DataEC50:  236nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM180437(US8772323, 1)
Affinity DataEC50:  660nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180438(US8772323, 2)
Affinity DataEC50:  787nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180439(US8772323, 3)
Affinity DataEC50:  82nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180440(US8772323, 4)
Affinity DataEC50:  596nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180441(US8772323, 5)
Affinity DataEC50:  243nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180442(US8772323, 6)
Affinity DataEC50:  1.70E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180443(US8772323, 7)
Affinity DataEC50:  892nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180444(US8772323, 8)
Affinity DataEC50:  874nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180445(US8772323, 9)
Affinity DataEC50:  834nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180446(US8772323, 10)
Affinity DataEC50:  365nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180447(US8772323, 11)
Affinity DataEC50: >1.00E+4nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180448(US8772323, 12)
Affinity DataEC50:  246nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180449(US8772323, 13)
Affinity DataEC50:  153nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180450(US8772323, 14)
Affinity DataEC50:  264nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180451(US8772323, 15)
Affinity DataEC50:  701nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180452(US8772323, 16)
Affinity DataEC50:  314nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180453(US8772323, 17)
Affinity DataEC50:  223nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180454(US8772323, 18)
Affinity DataEC50:  153nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180455(US8772323, 19)
Affinity DataEC50:  469nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180456(US8772323, 20)
Affinity DataEC50:  157nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180457(US8772323, 21)
Affinity DataEC50: >1.00E+4nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180458(US8772323, 22)
Affinity DataEC50:  1.75E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180459(US8772323, 23)
Affinity DataEC50:  1.35E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180460(US8772323, 24)
Affinity DataEC50:  5.10E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180461(US8772323, 25)
Affinity DataEC50:  2.37E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180462(US8772323, 26)
Affinity DataEC50:  166nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180463(US8772323, 27)
Affinity DataEC50:  444nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180464(US8772323, 28)
Affinity DataEC50:  213nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180466(US8772323, 29)
Affinity DataEC50:  181nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180467(US8772323, 30)
Affinity DataEC50: >1.00E+4nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180468(US8772323, 31)
Affinity DataEC50:  66nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180469(US8772323, 32)
Affinity DataEC50:  869nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180470(US8772323, 33)
Affinity DataEC50:  70nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180471(US8772323, 34)
Affinity DataEC50:  193nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180472(US8772323, 35)
Affinity DataEC50:  148nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180473(US8772323, 36)
Affinity DataEC50:  58nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180474(US8772323, 37)
Affinity DataEC50:  636nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180475(US8772323, 38)
Affinity DataEC50:  890nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180476(US8772323, 39)
Affinity DataEC50:  329nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180478(US8772323, 40)
Affinity DataEC50:  275nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180479(US8772323, 41)
Affinity DataEC50:  1.52E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180480(US8772323, 42)
Affinity DataEC50:  4.18E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180481(US8772323, 43)
Affinity DataEC50:  1.08E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180482(US8772323, 44)
Affinity DataEC50:  1.09E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180483(US8772323, 45)
Affinity DataEC50:  807nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180484(US8772323, 46)
Affinity DataEC50:  345nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180485(US8772323, 47)
Affinity DataEC50:  226nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM180486(US8772323, 48)
Affinity DataEC50:  348nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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