Report error Found 259 Enz. Inhib. hit(s) with Target = 'Gastrin-releasing peptide receptor'
Affinity DataEC50: 1.91E+4nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 84nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 41nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.22E+4nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Effective concentration required against gastrin releasing peptide receptor (GRP-R) in CHO cells by using FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0600nMAssay Description:Agonist activity at recombinant gastrin releasing peptide receptor expressed in baculovirus-transduced HEK293 cells assessed as intracellular calcium...More data for this Ligand-Target Pair
Affinity DataEC50: 0.258nMAssay Description:Displacement of 125I[Tyr4]-bombesin from GRPR expressed in human PC3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.373nMAssay Description:Displacement of 125I[Tyr4]-bombesin from GRPR expressed in human PC3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0380nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0790nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I-Tyr4]bombesin from GRPR (unknown origin) expressed in human PC3 cells after 45 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.650nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 1.24nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.45nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
