Compile Data Set for Download or QSAR
Report error Found 277 Enz. Inhib. hit(s) with Target = 'Galanin receptor type 2'
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM392076(US10301272, Example 7/9)
Affinity DataIC50: 0.190nMAssay Description:Displacement of [125I]-endothelin-1 from human recombinant GAL2 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2020
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85164(Galanin (1-29), rat)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85169(Galanin [D-Trp2], porcine | Galanin (1-29), porcin...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85164(Galanin (1-29), rat)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50307256(Gal(1-13)-Std I | CHEMBL604373 | GWTLNSAGYLLGPrPKP...)
Affinity DataKi:  0.600nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85172(CAS_112747-70-3 | Galanin (1-15))
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  0.850nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  0.900nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKd:  1nMAssay Description:Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | NSC_3043476 | Galantide (M15))
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  1.05nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85073(CAS_3043476 | NSC_3043476 | Galantide (M15))
Affinity DataKi:  1.07nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  1.10nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  1.11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  1.17nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin rat | Galanin (1-19), rat)
Affinity DataKi:  1.35nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50307255(GWTLNSAGYLLGPRHYINLITRQRY-CONH2 | CHEMBL592413)
Affinity DataKi:  1.40nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85168(M32)
Affinity DataKi:  1.45nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85164(Galanin (1-29), rat)
Affinity DataKi:  1.48nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  1.5nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85200(Galanin rat | Galanin (1-19), rat)
Affinity DataKi:  1.62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50307252(WTLNSAGYLL-CONH2 | CHEMBL578710)
Affinity DataKi:  1.70nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50273368(WTLNSAGYLL | CHEMBL506210)
Affinity DataKd:  1.80nMAssay Description:Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  1.80nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85069(Galanin Porcine 2-29 | Galanin (2-29), rat)
Affinity DataKi:  1.92nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/2/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  1.95nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273367(Galanin (1-16), rat | Galanin (1-16), porcine | CH...)
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKd:  2nMAssay Description:Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50273366(GWTLNSAGYLLGPHAVGNHRSFSDKNGLT | CHEMBL499179)
Affinity DataKd:  2.30nMAssay Description:Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  2.34nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50: 2.60nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2018
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273367(Galanin (1-16), rat | Galanin (1-16), porcine | CH...)
Affinity DataKi:  2.75nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  2.88nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2012
Entry Details Article
PubMed
TargetGalanin receptor type 2(Human)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM85069(Galanin Porcine 2-29 | Galanin (2-29), rat)
Affinity DataKi:  2.88nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
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