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Report error Found 137 Enz. Inhib. hit(s) with Target = 'Galanin receptor type 1' Sort by
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273368(WTLNSAGYLL | CHEMBL506210)
Affinity DataKd:  879nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKd:  0.300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKd:  0.100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273372(galmic | CHEMBL503924)
Affinity DataKd:  3.40E+4nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273366(GWTLNSAGYLLGPHAVGNHRSFSDKNGLT | CHEMBL499179)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273367(Galanin (1-16), rat | Galanin (1-16), porcine | CH...)
Affinity DataKd:  3.20nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50423646(Galnon | CHEMBL2309599)
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)
Affinity DataIC50: 0.0790nMAssay Description:Displacement of [125I]galanin from human recombinant GAL1 receptor expressed in HEK293 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2018
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50: 0.770nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50149871((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256665((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256666((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...)
Affinity DataIC50: 10.2nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256705((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...)
Affinity DataIC50: 11.1nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256704((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...)
Affinity DataIC50: 11.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256664((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...)
Affinity DataIC50: 20.4nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256706((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...)
Affinity DataIC50: 29.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50256746((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...)
Affinity DataIC50: 94.6nMAssay Description:Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358662(CHEMBL1922003)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358673(CHEMBL1922025)
Affinity DataIC50: 2.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358659(CHEMBL1922000)
Affinity DataIC50: 3.35E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358670(CHEMBL1922022)
Affinity DataIC50: 3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358669(CHEMBL1922021)
Affinity DataIC50: 3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358660(CHEMBL1922001)
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358653(CHEMBL1921993)
Affinity DataIC50: 4.60E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358655(CHEMBL1921996)
Affinity DataIC50: 5.03E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358667(CHEMBL1922016)
Affinity DataIC50: 5.48E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358657(CHEMBL1921998)
Affinity DataIC50: 5.62E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358656(CHEMBL1921997)
Affinity DataIC50: 5.93E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358661(CHEMBL1922002)
Affinity DataIC50: 6.32E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358651(CHEMBL1921991)
Affinity DataIC50: 6.77E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358668(CHEMBL1922019)
Affinity DataIC50: 6.78E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358671(CHEMBL1922023)
Affinity DataIC50: 6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358658(CHEMBL1921999)
Affinity DataIC50: 6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358650(CHEMBL1921989)
Affinity DataIC50: 6.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358648(CHEMBL1921902)
Affinity DataIC50: 8.59E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358652(CHEMBL1921992)
Affinity DataIC50: 1.28E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358672(CHEMBL1922024)
Affinity DataIC50: 1.60E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358654(CHEMBL1921995)
Affinity DataIC50: 2.75E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50358649(CHEMBL1921903)
Affinity DataIC50: 3.49E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Rat)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307256(Gal(1-13)-Std I | CHEMBL604373 | GWTLNSAGYLLGPrPKP...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | M35 | Galanin (1-13)-bradikinin(2-9...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
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