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Report error Found 31 Enz. Inhib. hit(s) with Target = 'Gag-Pro polyprotein'
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371707(KNI-10221 | CHEMBL272710)
Affinity DataIC50: 84nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371728(KNI-10166 | CHEMBL271706)
Affinity DataIC50: 88nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371720(KNI-10192 | CHEMBL272280)
Affinity DataIC50: 95nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371718(KNI-10220 | CHEMBL271878)
Affinity DataIC50: 101nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371725(KNI-10199 | CHEMBL403182)
Affinity DataIC50: 102nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371706(CHEMBL404702)
Affinity DataIC50: 103nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50242888(KNI-10516 | (R)-3-((2S,3S)-3-((S)-2-((S)-2-acetami...)
Affinity DataIC50: 107nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371712(KNI-10600 | CHEMBL256022)
Affinity DataIC50: 113nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371721(KNI-10197 | CHEMBL403770)
Affinity DataIC50: 123nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371715(KNI-10496 | CHEMBL256587)
Affinity DataIC50: 131nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371705(KNI-10455 | CHEMBL401718)
Affinity DataIC50: 140nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371717(KNI-10247 | CHEMBL404836)
Affinity DataIC50: 144nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371724(KNI-10194 | CHEMBL272920)
Affinity DataIC50: 145nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371713(KNI-10592 | CHEMBL271454)
Affinity DataIC50: 146nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371729(CHEMBL436816)
Affinity DataIC50: 152nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50227057((S)-2-((S)-2-((S)-2-((S)-1-((2S,3S)-3-((S)-2-((S)-...)
Affinity DataIC50: 159nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371719(KNI-10191 | CHEMBL256385)
Affinity DataIC50: 159nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371708(KNI-10193 | CHEMBL257647)
Affinity DataIC50: 160nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371722(KNI-10196 | CHEMBL402525)
Affinity DataIC50: 180nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371723(KNI-10188 | CHEMBL401814)
Affinity DataIC50: 180nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371714(KNI-10502 | CHEMBL256588)
Affinity DataIC50: 193nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371710(KNI-10198 | CHEMBL256386)
Affinity DataIC50: 201nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371726(KNI-10168 | CHEMBL257649)
Affinity DataIC50: 249nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371709(KNI-10195 | CHEMBL272494)
Affinity DataIC50: 320nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371711(KNI-10127 | CHEMBL233649)
Affinity DataIC50: 353nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371716(KNI-10401 | CHEMBL258157)
Affinity DataIC50: 473nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50371727(KNI-10167 | CHEMBL430094)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HTLV1 protease L40I mutant expressed in Escherichia coli BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50155805(H-Pro-Gln-Val-Apns-Dmt-Val-Met-His-OH | CHEMBL4156...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibitory binding affinity towards synthesized human T-cell leukemia virus type I (HTLV-1) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50155805(H-Pro-Gln-Val-Apns-Dmt-Val-Met-His-OH | CHEMBL4156...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibitory binding affinity towards recombinant human T-cell leukemia virus type I (HTLV-1) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataKi:  1.46E+4nMAssay Description:Inhibitory binding affinity towards recombinant human T-cell leukemia virus type I (HTLV-1) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGag-Pro polyprotein(HTLV-1)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataKi:  3.65E+4nMAssay Description:Inhibitory binding affinity towards synthesized human T-cell leukemia virus type I (HTLV-1) proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed