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Report error Found 342 Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 1'
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439404(CHEMBL2420539)
Affinity DataEC50:  3.60E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM95731(cid_4101833 | SMR000244241 | 2-(4-chlorophenyl)-N-...)
Affinity DataEC50:  2.30E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439405(CHEMBL2420538)
Affinity DataEC50:  3.30E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439402(CHEMBL2420537)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439403(CHEMBL1558022)
Affinity DataEC50:  1.10E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437983(CHEMBL2409106)
Affinity DataEC50:  160nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50115223(1-(5-Methyl-2-phenyl-2H-pyrazol-3-yl)-3-phenyl-ure...)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50241582(cid_25075 | CHEMBL451532 | cid_442428 | (S)-7-((2S...)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of recombinant human GIRK1/2 expressed in Xenopus oocytes by two-electrode voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439406(CHEMBL2420536)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439407(CHEMBL2420535)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439408(CHEMBL2420534)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439409(CHEMBL2420533)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439410(CHEMBL2420532)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439411(CHEMBL2420531)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439412(CHEMBL2420530)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439413(CHEMBL2420529)
Affinity DataEC50:  5.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439414(CHEMBL2420550)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439415(CHEMBL2420549)
Affinity DataEC50:  3.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439416(CHEMBL2420548)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439417(CHEMBL2420547)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439418(CHEMBL2420546)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439419(CHEMBL2420545)
Affinity DataEC50:  1.10E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439420(CHEMBL2420544)
Affinity DataEC50:  3.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439421(CHEMBL2420543)
Affinity DataEC50:  1.70E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439422(CHEMBL2420542)
Affinity DataEC50:  2.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439423(CHEMBL2420541)
Affinity DataEC50:  3.30E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439424(CHEMBL2420540)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50437968(CHEMBL2409134)
Affinity DataEC50:  3.50E+3nMAssay Description:Activation of GIRK1/4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437983(CHEMBL2409106)
Affinity DataEC50:  160nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50115223(1-(5-Methyl-2-phenyl-2H-pyrazol-3-yl)-3-phenyl-ure...)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437968(CHEMBL2409134)
Affinity DataEC50:  1.70E+3nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437969(CHEMBL2409133)
Affinity DataEC50:  470nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437970(CHEMBL2409132)
Affinity DataEC50:  210nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437971(CHEMBL2409131)
Affinity DataEC50:  350nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437972(CHEMBL2409130)
Affinity DataEC50:  570nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437973(CHEMBL2409129)
Affinity DataEC50:  380nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437974(CHEMBL2409128)
Affinity DataEC50:  530nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437975(CHEMBL2409127)
Affinity DataEC50:  340nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437976(CHEMBL2409120)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437963(CHEMBL2409117)
Affinity DataEC50:  3.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437965(CHEMBL2409115)
Affinity DataEC50:  3.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437977(CHEMBL2409113)
Affinity DataEC50:  410nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437967(CHEMBL2409112)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437978(CHEMBL2409111)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437979(CHEMBL2409110)
Affinity DataEC50:  70nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437980(CHEMBL2409109)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437981(CHEMBL2409108)
Affinity DataEC50:  190nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50437982(CHEMBL2409107)
Affinity DataEC50:  460nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataEC50:  0.0614nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetG protein-activated inward rectifier potassium channel 1(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | TCMDC-12...)
Affinity DataEC50:  1.49nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
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