Compile Data Set for Download or QSAR
Report error Found 670 Enz. Inhib. hit(s) with Target = 'Fatty acid-binding protein 5'
TargetFatty acid-binding protein 5(Mouse)
Case Western Reserve University School of Medicine

LigandPNGBDBM60927(ANS | BDBM50126831 | 1-anilinonaphthalene-8-sulfon...)
Affinity DataKd:  70nMAssay Description:The method entails two steps [Lin et al., Biochemistry, 38:185-190]. In the first step, the Kd for association of FABP5 with the fluorescent lipid pr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5-ANS(Mouse)
Case Western Reserve University School of Medicine

LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataKd:  100nMAssay Description:The method entails two steps [Lin et al., Biochemistry, 38:185-190]. In the first step, the Kd for association of FABP5 with the fluorescent lipid pr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5-ANS(Mouse)
Case Western Reserve University School of Medicine

LigandPNGBDBM22319([1-14C]Arachidonic acid | (5Z,8Z,11Z,14Z)-icosa-5,...)
Affinity DataKd:  42.1nMAssay Description:The method entails two steps [Lin et al., Biochemistry, 38:185-190]. In the first step, the Kd for association of FABP5 with the fluorescent lipid pr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM60927(ANS | BDBM50126831 | 1-anilinonaphthalene-8-sulfon...)
Affinity DataKd:  6.57E+3nMpH: 8.2 T: 2°CAssay Description:In brief, both wild-type and mutant hFABP5 were expressed and purified to homogeneity as described above and dialyzed in PBS (pH 8.2). Binding affini...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM60927(ANS | BDBM50126831 | 1-anilinonaphthalene-8-sulfon...)
Affinity DataKd:  1.26E+4nMpH: 8.2 T: 2°CAssay Description:In brief, both wild-type and mutant hFABP5 were expressed and purified to homogeneity as described above and dialyzed in PBS (pH 8.2). Binding affini...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5 [M35A,L60A](Human)
Emory University

LigandPNGBDBM60927(ANS | BDBM50126831 | 1-anilinonaphthalene-8-sulfon...)
Affinity DataKd:  6.10E+3nMpH: 8.2 T: 2°CAssay Description:In brief, both wild-type and mutant hFABP5 were expressed and purified to homogeneity as described above and dialyzed in PBS (pH 8.2). Binding affini...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM50152850(1-HEXYLDECANOIC ACID | Hexadecanoic acid anion | H...)
Affinity DataKd:  802nMAssay Description:Binding affinity to human kFABPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM50574778(CHEMBL4851660)
Affinity DataKd:  1.05E+5nMAssay Description:Binding affinity to FABP5 (unknown origin) by microscale thermophoresis analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM50468360(CHEMBL4280900)
Affinity DataKd:  2.79E+6nMAssay Description:Binding affinity to FABP5 (unknown origin) by microscale thermophoresis analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM50574783(CHEMBL4864312)
Affinity DataKd:  1.41E+4nMAssay Description:Binding affinity to FABP5 (unknown origin) by microscale thermophoresis analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312342(US9604977, Example 88 | 2-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312347(US9604977, Example 93 | 3-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312356(US9604977, Example 102 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312447(US9604977, Example 193 | 2-[6-Ethyl-3-(4-methyl-th...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312420(US9604977, Example 166 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 13nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312421(US9604977, Example 167 | 2-[(S)-3-(3-Cyclopropyl-[...)
Affinity DataIC50: 13nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234709(US9353102, 4.15)
Affinity DataIC50: 16nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312422(US9604977, Example 168 | 2-[(R)-3-(3-Cyclopropyl-[...)
Affinity DataIC50: 18nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312472(US9604977, Example 218 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 19nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312313(US9604977, Example 61 | 2-[3-(3-Trifluoromethyl-[1...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312330(US9604977, Example 77 | 2-[4,4-Dimethyl-3-(3-methy...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312338(US9604977, Example 85 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312340(US9604977, Example 86 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312346(US9604977, Example 92 | 2-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312363(US9604977, Example 109 | (−)-2-[3-(3-Cyclopr...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312401(US9604977, Example 147 | 2-[6,6-Difluoro-3-(3-trif...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312405(US9604977, Example 151 | 2-[6,6-Difluoro-3-(4-meth...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM50615292(CHEMBL5278217)
Affinity DataIC50: 20nMAssay Description:Inhibition of human FABP5More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234703(US9353102, 4.9)
Affinity DataIC50: 22nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234707(US9353102, 4.13)
Affinity DataIC50: 22nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312442(US9604977, Example 188 | 2-[3-(4-Methyl-thiazol-2-...)
Affinity DataIC50: 22nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234674(US9353102, 3.3)
Affinity DataIC50: 30nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234678(US9353102, 4.2)
Affinity DataIC50: 30nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234681(US9353102, 4.5)
Affinity DataIC50: 30nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234704(US9353102, 4.10)
Affinity DataIC50: 30nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM234682(US9353102, 5)
Affinity DataIC50: 30nMpH: 7.5Assay Description:Stock DMSO solutions (1.8 mM) of compounds were serially diluted 3-fold for ten concentrations with 100% DMSO (50 μM to 0.003 μM final comp...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312314(US9604977, Example 62 | 3-[3-(3-Trifluoromethyl-[1...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312333(US9604977, Example 80 | 3-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312341(US9604977, Example 87 | 3-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312357(US9604977, Example 103 | 3-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312372(US9604977, Example 118 | 2-[5-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312378(US9604977, Example 124 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312380(US9604977, Example 126 | 2-[3-(3-Trifluoromethyl-[...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312382(US9604977, Example 128 | 3-[3-(3-Trifluoromethyl-[...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312386(US9604977, Example 132 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312398(US9604977, Example 144 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312404(US9604977, Example 150 | 2-[6,6-Difluoro-3-(4-meth...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312460(US9604977, Example 206 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM312485(US9604977, Example 231 | 2-[6,6-Difluoro-3-(4-isop...)
Affinity DataIC50: 30nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetFatty acid-binding protein 5(Human)
Emory University

LigandPNGBDBM50615291(CHEMBL5287082)
Affinity DataIC50: 30nMAssay Description:Inhibition of human FABP5More data for this Ligand-Target Pair
In DepthDetails
PubMed
Displayed 1 to 50 (of 670 total ) | Next | Last >>
Jump to: