Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with Target = 'Eukaryotic translation initiation factor 2 subunit 1'
LigandPNGBDBM50570964(CHEMBL4857782)
Affinity DataIC50: 9nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50570960(CHEMBL4858308)
Affinity DataIC50: 18nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570963(CHEMBL4848143)
Affinity DataIC50: 23nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570956(CHEMBL4869882)
Affinity DataIC50: 27nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570941(CHEMBL4862478)
Affinity DataIC50: 33nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570958(CHEMBL4853221)
Affinity DataIC50: 40nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570972(CHEMBL4848359)
Affinity DataIC50: 40nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570966(CHEMBL4861671)
Affinity DataIC50: 42nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570955(CHEMBL4863698)
Affinity DataIC50: 45nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570952(CHEMBL4870100)
Affinity DataIC50: 49nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570959(CHEMBL4870780)
Affinity DataIC50: 54nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570953(CHEMBL4875875)
Affinity DataIC50: 58nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570962(CHEMBL4851480)
Affinity DataIC50: 72nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570957(CHEMBL4876496)
Affinity DataIC50: 114nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570968(CHEMBL4854504)
Affinity DataIC50: 181nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570942(CHEMBL4852735)
Affinity DataIC50: 187nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570943(CHEMBL4870495)
Affinity DataIC50: 198nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570944(CHEMBL4866245)
Affinity DataIC50: 307nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570961(CHEMBL4846663)
Affinity DataIC50: 313nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570965(CHEMBL4870565)
Affinity DataIC50: 366nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570969(CHEMBL4849149)
Affinity DataIC50: 638nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570948(CHEMBL4868021)
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570954(CHEMBL4876223)
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570946(CHEMBL4853233)
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570949(CHEMBL4848921)
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570947(CHEMBL4854364)
Affinity DataIC50: 3.34E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570970(CHEMBL4858598)
Affinity DataIC50: 4.03E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570967(CHEMBL4878188)
Affinity DataIC50: 7.65E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570945(CHEMBL4856844)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50570971(CHEMBL4853611)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed