Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor [S768I]'
TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557850(US11365189, Ex. No. 4 | 6-((1-acryloylpiperidin-4-...)
Affinity DataIC50: 0.130nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557852(US11365189, Ex. No. 6 | 1-(3-((4-((3,4-dichloro-2-...)
Affinity DataIC50: 0.350nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557849(US11365189, Ex. No. 3 | 1-(3-((4-((3,4-dichlorophe...)
Affinity DataIC50: 0.510nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM50468247(HM 781-36B | HM-781-36B | NOV-120101 | Poziotinib ...)
Affinity DataIC50: 0.910nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557865(US11365189, Ex. No. 25 | 1-(4-((4-((3,4-dichloro- ...)
Affinity DataIC50: 2nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557851(US11365189, Ex. No. 5 | 1-(3-((4-((2,4-dichlorophe...)
Affinity DataIC50: 2.5nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557875(US11365189, Ex. No. 41 | 1-(3-((7-methoxy-4- (phen...)
Affinity DataIC50: 2.90nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557870(US11365189, Ex. No. 32 | 1-(3-((4-((3,4-dichloro-2...)
Affinity DataIC50: 3.90nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557858(US11365189, Ex. No. 14 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 4nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557868(US11365189, Ex. No. 30 | 1-(3-((4-((4-bromo-3- chl...)
Affinity DataIC50: 4.80nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557846(US11365189, Ex. No. 1 | 1-(4-((4-((2,4-dichlorophe...)
Affinity DataIC50: 5nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557872(US11365189, Ex. No. 37 | 1-(4-((4-((4-bromo-3- chl...)
Affinity DataIC50: 5nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557867(US11365189, Ex. No. 29 | 1-(4-((7-methoxy-4-((3- (...)
Affinity DataIC50: 6.5nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557898(US11365189, Ex. No. 48 | 1-(3-((4-((3,4-dichloro- ...)
Affinity DataIC50: 6.60nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557869(US11365189, Ex. No. 31 | 1-(3-((4-((3-cyclopropyl-...)
Affinity DataIC50: 8.10nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557888(US11365189, Ex. No. 24 | 1-(3-((4-((4-bromo-3- chl...)
Affinity DataIC50: 10nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557854(US11365189, Ex. No. 9)
Affinity DataIC50: 11nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557899(US11365189, Ex. No. 51 | 1-(3-((4-((4-chloro-3- (o...)
Affinity DataIC50: 14nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557890(US11365189, Ex. No. 28 | 1-(4-((4-((3-cyclopropyl-...)
Affinity DataIC50: 15nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557861(US11365189, Ex. No. 16 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 19nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557877(US11365189, Ex. No. 49 | 1-(3-((7-methoxy-4-((3- (...)
Affinity DataIC50: 20nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557866(US11365189, Ex. No. 27 | 1-(3-((7-methoxy-4-((3- (...)
Affinity DataIC50: 20nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557873(US11365189, Ex. No. 39 | 1-(4-((7-methoxy-4- (phen...)
Affinity DataIC50: 33nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557878(US11365189, Ex. No. 50 | 1-(3-((7-methoxy-4- (phen...)
Affinity DataIC50: 34nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557881(US11365189, Ex. No. 99 | 1-(3-((4-((4-bromo-3- chl...)
Affinity DataIC50: 35nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557848(US11365189, Ex. No. 2 | 1-(3-((4-((2,4-dichlorophe...)
Affinity DataIC50: 48nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557886(US11365189, Ex. No. 22 | 1-(4-((4-((4-chloro-3- (o...)
Affinity DataIC50: 53nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557860(US11365189, Ex. No. 15 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 66nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557897(US11365189, Ex. No. 47 | 1-(3-((4-((4-chloro-3- (o...)
Affinity DataIC50: 66nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557883(US11365189, Ex. No. 18 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 67nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557880(US11365189, Ex. No. 54 | 1-(3-((4-((4-chloro-3- (h...)
Affinity DataIC50: 69nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557855(US11365189, Ex. No. 11 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 81nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557882(US11365189, Ex. No. 17 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 95nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557871(US11365189, Ex. No. 35 | 1-(3-((7-methoxy-4-((4- (...)
Affinity DataIC50: 100nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557887(US11365189, Ex. No. 23 | 1-(4-((4-((3-chloro-4- (t...)
Affinity DataIC50: 110nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557892(US11365189, Ex. No. 34 | 1-(4-((4-((4-chloro-3- (h...)
Affinity DataIC50: 110nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557874(US11365189, Ex. No. 40 | 1-(3-((4-((2,4-dichloro- ...)
Affinity DataIC50: 130nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557876(US11365189, Ex. No. 43 | 1-(3-((4-((3-chloro-4- (t...)
Affinity DataIC50: 130nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557901(US11365189, Ex. No. 55 | 1-(3-((4-((4-chloro-3- (h...)
Affinity DataIC50: 210nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557900(US11365189, Ex. No. 52 | 1-(4-((7-methoxy-4-((4- (...)
Affinity DataIC50: 220nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557895(US11365189, Ex. No. 44 | 1-(3-((4-((3-cyclopropyl-...)
Affinity DataIC50: 250nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557903(US11365189, Ex. No. 57 | 1-(3-((4-((3-(hydroxy- me...)
Affinity DataIC50: 490nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557894(US11365189, Ex. No. 38 | 1-(3-((4-((3-chloro-4- (t...)
Affinity DataIC50: 510nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557856(US11365189, Ex. No. 12 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 650nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557885(US11365189, Ex. No. 21 | 1-(4-((4-((3-(hydroxy- me...)
Affinity DataIC50: 740nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557896(US11365189, Ex. No. 45 | 1-(3-((7-methoxy-4-((4- (...)
Affinity DataIC50: 1.00E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557908(US11365189, Ex. No. 93 | 1-(3-((4-((2,4-dichloro- ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557864(US11365189, Ex. No. 20 | 6-((1-acryloylpiperidin-4...)
Affinity DataIC50: 1.80E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557879(US11365189, Ex. No. 53 | 1-(3-((7-methoxy-4-((1- m...)
Affinity DataIC50: 2.20E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [S768I](Human)
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM557907(US11365189, Ex. No. 62 | 1-(3-((4-((4-chloro-3-cyc...)
Affinity DataIC50: 2.50E+3nMAssay Description:Cell viability was determined using the Cell Titer Glo assay (Promega) as previously described. Briefly, 2000-3000 cells per well were plated in 384-...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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