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Report error Found 416 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor [L858R,T790M,C797S]'
TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM561454(US11390625, Compound 34 | US11390625, Example 34)
Affinity DataIC50: 0.160nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM561456(US11390625, Compound 44 | US11390625, Example 44)
Affinity DataIC50: 0.210nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM495017(US10994015, Example 313 | US10994015, Example 314)
Affinity DataIC50: 0.260nMAssay Description:All compounds and PROTACs were serially diluted in three-fold increments using 100% DMSO, followed by an intermediate 10-fold dilution using Buffer A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM561455(US11390625, Compound 41 | US11390625, Example 41)
Affinity DataIC50: 0.260nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM495012(US10994015, Example 308)
Affinity DataIC50: 0.270nMAssay Description:All compounds and PROTACs were serially diluted in three-fold increments using 100% DMSO, followed by an intermediate 10-fold dilution using Buffer A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM495016(US10994015, Example 312)
Affinity DataIC50: 0.350nMAssay Description:All compounds and PROTACs were serially diluted in three-fold increments using 100% DMSO, followed by an intermediate 10-fold dilution using Buffer A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM495019(US10994015, Example 319)
Affinity DataIC50: 0.800nMAssay Description:All compounds and PROTACs were serially diluted in three-fold increments using 100% DMSO, followed by an intermediate 10-fold dilution using Buffer A...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649309(US20240034743, Compound 1)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649310(US20240034743, Compound 2)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649311(US20240034743, Compound 3)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649312(US20240034743, Compound 4)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649313(US20240034743, Compound 5)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649314(US20240034743, Compound 6)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649315(US20240034743, Compound 7)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649316(US20240034743, Compound 8)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649317(US20240034743, Compound 9)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649318(US20240034743, Compound 10)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649319(US20240034743, Compound 11)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649320(US20240034743, Compound 12)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649321(US20240034743, Compound 13)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649322(US20240034743, Compound 14)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649323(US20240034743, Compound 15)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649324(US20240034743, Compound 16)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649327(US20240034743, Compound 19)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649328(US20240034743, Compound 20)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649329(US20240034743, Compound 21)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649332(US20240034743, Compound 24)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649333(US20240034743, Compound 25)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649334(US20240034743, Compound 26)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649335(US20240034743, Compound 78 | US20240034743, Compou...)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649336(US20240034743, Compound 28)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649337(US20240034743, Compound 29)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649338(US20240034743, Compound 30)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649339(US20240034743, Compound 31)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649340(US20240034743, Compound 32)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649341(US20240034743, Compound 33)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649343(US20240034743, Compound 35)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649344(US20240034743, Compound 36)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649345(US20240034743, Compound 37)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649346(US20240034743, Compound 38)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649347(US20240034743, Compound 39)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649348(US20240034743, Compound 40)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649349(US20240034743, Compound 41)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649350(US20240034743, Compound 42)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649351(US20240034743, Compound 43)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649352(US20240034743, Compound 44)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649353(US20240034743, Compound 100 | US20240034743, Compo...)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649354(US20240034743, Compound 46)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649355(US20240034743, Compound 47)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetEpidermal growth factor receptor [L858R,T790M,C797S](Human)
Chia Tai Tianqing Pharmaceutical Group

US Patent
LigandPNGBDBM649356(US20240034743, Compound 48)
Affinity DataIC50: 1nMAssay Description:TBDMore data for this Ligand-Target Pair
In DepthDetails
US Patent

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