Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with Target = 'Endothelin receptor type B/1 receptor'
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045239(Ac-D-Dip-Leu-Asp-Ile-Ile-Trp | Ac-D-Dip-Leu-Asp-Il...)
Affinity DataIC50: 25nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368647(CHEMBL1788127)
Affinity DataIC50: 40nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045230(Ac-D-Trp-Leu-Asp-Ile-Ile-Trp | CHEMBL313382)
Affinity DataIC50: 130nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045244(Ac-D-Phe-D-Phe-Asp-Ile-Ile-Trp | (S)-3-[(S)-2-((R)...)
Affinity DataIC50: 330nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045240(Ac-D-Phe-Leu-Phe-Ile-Ile-Trp | (S)-2-[(S)-2-((2S,5...)
Affinity DataIC50: 380nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001219(CHEMBL85341 | 3-{2-[2-Acetylamino-3-(4-hydroxy-phe...)
Affinity DataIC50: 400nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045262(Ac-D-Phe-Ala-Asp-Ile-Ile-Trp | CHEMBL406279)
Affinity DataIC50: 420nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045227(Ac-D-Phe-Orn-Asp-Ile-Ile-Trp | (S)-3-[2-((R)-2-Ace...)
Affinity DataIC50: 680nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001217(CHEMBL86814 | 3-[2-(2-Acetylamino-3-phenyl-propion...)
Affinity DataIC50: 740nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045243(Ac-D-Phe-Glu-Asp-Ile-Trp | CHEMBL313056)
Affinity DataIC50: 740nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001221(CHEMBL315047 | 3-[2-(2-Acetylamino-3-naphthalen-2-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045237(Ac-D-Phe-Leu-Asp-Ala-Ile-Trp | CHEMBL87243)
Affinity DataIC50: 1.61E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045251(Ac-D-Phe-Asp-Ile-Ile-Trp | 3-((R)-2-Acetylamino-3-...)
Affinity DataIC50: 2.15E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045250(Ac-D-Phe-Leu-Asp-Ile-Ile-Bta | CHEMBL315780)
Affinity DataIC50: 3.80E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000566((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 4.10E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001218(CHEMBL438194 | 3-[2-(2-Acetylamino-3-biphenyl-4-yl...)
Affinity DataIC50: 4.40E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000566((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 4.50E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50231133(CHEMBL262166)
Affinity DataIC50: 5.20E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045225(Ac-D-Phe-Leu-Asp-Ile-Ala-Trp | CHEMBL86737)
Affinity DataIC50: 6.83E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045232(Ac-D-Phe-Leu-Asp-Glu-Ile-Trp | CHEMBL431874)
Affinity DataIC50: 9.00E+3nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045260(Ac-D-Phe-Leu-Lys-Ile-Ile-Trp | CHEMBL431218)
Affinity DataIC50: 1.20E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045265(D-Phe-Leu-Asp-Ile-Ile-Trp | CHEMBL315328)
Affinity DataIC50: 1.24E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50231134(CHEMBL2370061)
Affinity DataIC50: 1.69E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045235((S)-3-[(R)-2-((1S,5S)-2-Acetylamino-3-phenyl-propi...)
Affinity DataIC50: 2.45E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50231136(CHEMBL2370073)
Affinity DataIC50: 3.70E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50231135(CHEMBL2114215)
Affinity DataIC50: 3.90E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50231137(CHEMBL2369145)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50231132(CHEMBL313122)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50045229(Ac-D-Phe-Leu-Asp-Lys-Ile-Trp | CHEMBL314239)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001214(CHEMBL432091 | 3-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataIC50: 5.80E+4nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50231138(CHEMBL3350293)
Affinity DataIC50: 1.69E+5nMAssay Description:Binding affinity against Endothelin receptor from rat heart ventricleMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000564(CHEMBL538475 | 2-[2-{[2-(Cyclohexanecarbonyl-amino...)
Affinity DataIC50: 2.30E+5nMAssay Description:Compound was evaluated for the Inhibition of the contractile response of Endothelin A receptor in rabbit thoracic aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndothelin receptor type B/1 receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50187377(N-(3-(4-(4-(cyclohexylmethylsulfonamido)butyl)pipe...)
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity to endothelin receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed